SCHEMBL211763

SCHEMBL211763

COc1ccc2nc(NC=O)sc2c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 12/20 0.64
RAB9A P51151 12/20 0.64
SMN1; SMN2 Q16637 8/20 0.64
HTT P42858 4/20 0.64
CYP1A2 P05177 1/20 0.64
CYP3A4 P08684 1/20 0.64
CYP2C19 P33261 1/20 0.64
DYRK1A Q13627 1/20 0.64
MEN1 O00255 9/20 0.63
KMT2A Q03164 9/20 0.63
MAPT P10636 9/20 0.63
NFKB1 P19838 4/20 0.60
NFKB2 Q00653 4/20 0.60
RELA Q04206 4/20 0.60
SCD O00767 5/20 0.60
ATAD2 Q6PL18 1/20 0.60
ALDH1A1 P00352 5/20 0.59
GAA P10253 2/20 0.59
CASP2 P42575 1/20 0.59
TSHR P16473 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10531725 0.85 NPC1 (0.63) NPC1RAB9ASMN1; SMN2HTTCYP1A2
SCHEMBL19597485 0.85 NPC1 (0.63) NPC1RAB9ASMN1; SMN2HTTCYP1A2
SCHEMBL10531711 0.85 NPC1 (0.63) NPC1RAB9ASMN1; SMN2HTTCYP1A2
SCHEMBL1307056 0.83 MAPT (0.82) NPC1RAB9ASMN1; SMN2HTTCYP1A2
SCHEMBL211725 0.82 DYRK1A (0.65) NPC1RAB9ASMN1; SMN2HTTCYP1A2
SCHEMBL8280120 0.81 NPC1 (0.70) NPC1RAB9ASMN1; SMN2HTTCYP1A2
SCHEMBL16317400 0.81 SCD (0.51) NPC1RAB9ASMN1; SMN2HTTCYP1A2
SCHEMBL2114859 0.80 NPC1 (0.68) NPC1RAB9ASMN1; SMN2HTTCYP1A2
SCHEMBL14189675 0.80 NPC1 (0.61) NPC1RAB9ASMN1; SMN2HTTDYRK1A
SCHEMBL10991640 0.80 NPC1 (0.57) NPC1RAB9ASMN1; SMN2HTTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088793-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2012-01-03 US disclosed
WO-2005092899-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2005-10-06 WO disclosed