SCHEMBL21177142

SCHEMBL21177142

COC(=O)c1cnc(Cc2cc(F)c3ncc(Cl)cc3c2)o1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 9/20 0.36
S1PR1 P21453 1/20 0.35
S1PR3 Q99500 1/20 0.35
TP53 P04637 1/20 0.33
MAP4K1 Q92918 1/20 0.33
MMEL1 Q495T6 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPT P10636 2/20 0.32
FAAH O00519 1/20 0.32
CES1 P23141 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21177567 0.86 KLKB1 (0.35) KLKB1MAP4K1MMEL1
SCHEMBL19780407 0.80 KLKB1 (0.42) KLKB1S1PR1S1PR3SMN1; SMN2
SCHEMBL19779879 0.80 KLKB1 (0.52) KLKB1MAP4K1ALDH1A1SMN1; SMN2
SCHEMBL21177781 0.78 KLKB1 (0.36) KLKB1S1PR1S1PR3TP53MAP4K1
SCHEMBL20531521 0.78 KLKB1 (0.43) KLKB1ALDH1A1MAPT
SCHEMBL21177362 0.78 KLKB1 (0.38) KLKB1MAP4K1ALDH1A1SMN1; SMN2
SCHEMBL21177169 0.78 KLKB1 (0.51) KLKB1MAP4K1
SCHEMBL17442513 0.78 KLKB1 (0.49) KLKB1MAP4K1
SCHEMBL21179410 0.77 HSP90AB1 (0.42) KLKB1L3MBTL1ALDH1A1SMN1; SMN2KMT2A
SCHEMBL21177545 0.76 KLKB1 (0.34) KLKB1MAP4K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019142053-A2 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHARMACEUTICALS, INC. (BB) 2019-07-25 WO disclosed
WO-2019142053-A2 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHARMACEUTICALS, INC. (BB) 2019-07-25 WO disclosed