SCHEMBL21177781

SCHEMBL21177781

CCOC(=O)c1oc(Cc2cc(F)c3ncc(Cl)cc3c2)nc1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 5/20 0.36
S1PR1 P21453 1/20 0.35
S1PR3 Q99500 1/20 0.35
MAP4K1 Q92918 1/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPT P10636 2/20 0.33
HSD17B10 Q99714 2/20 0.33
MAOB P27338 2/20 0.33
GAA P10253 1/20 0.33
NPC1 O15118 1/20 0.33
TP53 P04637 1/20 0.33
XBP1 P17861 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TLR9 Q9NR96 1/20 0.33
BRAF P15056 1/20 0.33
EIF2AK3 Q9NZJ5 1/20 0.33
KMT2A Q03164 2/20 0.32
ALOX5 P09917 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21177362 0.89 KLKB1 (0.38) KLKB1MAP4K1ALDH1A1SMN1; SMN2
SCHEMBL21177327 0.89 S1PR1 (0.37) KLKB1S1PR1S1PR3ALDH1A1MAPT
SCHEMBL19780407 0.84 KLKB1 (0.42) KLKB1S1PR1S1PR3MAPK1NPSR1
SCHEMBL21179351 0.82 KLKB1 (0.51) KLKB1MAP4K1
SCHEMBL21177161 0.81 KLKB1 (0.42) KLKB1MAP4K1ALDH1A1MAPK1NPSR1
SCHEMBL21190192 0.78 ALOX15 (0.37) KLKB1S1PR1S1PR3ALDH1A1MAPT
SCHEMBL21177545 0.78 KLKB1 (0.34) KLKB1MAP4K1
SCHEMBL21177320 0.78 KLKB1 (0.33) KLKB1MAP4K1
SCHEMBL21177142 0.78 KLKB1 (0.36) KLKB1S1PR1S1PR3MAP4K1ALDH1A1
SCHEMBL21177623 0.78 KLKB1 (0.33) KLKB1MAP4K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019142053-A2 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHARMACEUTICALS, INC. (BB) 2019-07-25 WO disclosed
WO-2019142053-A2 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHARMACEUTICALS, INC. (BB) 2019-07-25 WO disclosed