SCHEMBL21180342

SCHEMBL21180342

O=C1CNCC(Cc2cccc(Br)c2)N1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 1/20 0.37
PARP1 P09874 2/20 0.37
PARP15 Q460N3 1/20 0.36
PARP10 Q53GL7 1/20 0.36
MAOB P27338 3/20 0.36
MAOA P21397 2/20 0.36
TAAR1 Q96RJ0 1/20 0.36
IDO1 P14902 2/20 0.35
AGXT P21549 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
FFAR1 O14842 1/20 0.34
PPARA Q07869 1/20 0.34
MMP2 P08253 2/20 0.34
GPR84 Q9NQS5 1/20 0.34
MMP1 P03956 1/20 0.34
MMP9 P14780 1/20 0.34
MMP12 P39900 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL682821 0.82 HDAC8 (0.45) CXCR4
SCHEMBL2088808 0.82 HDAC8 (0.45) CXCR4
SCHEMBL682465 0.82 HDAC8 (0.45) CXCR4
SCHEMBL30595821 0.77 TAAR1 (0.38) PARP1MAOBMAOATAAR1IDO1
SCHEMBL21180314 0.77 TAAR1 (0.38) PARP1MAOBMAOATAAR1IDO1
SCHEMBL1177121 0.76 MAOB (0.36) PARP1PARP15PARP10MAOBMAOA
SCHEMBL21187235 0.76 CXCR4 (0.39) CXCR4GPR84
SCHEMBL29452904 0.76 CXCR4 (0.39) CXCR4GPR84
SCHEMBL3878053 0.73 GAA (0.41) CXCR4
SCHEMBL18577318 0.73 CMA1 (0.39) CXCR4MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108250058-B PPAR agonists and their use in the treatment of Alzheimer's disease and other diseases 上海怡立舍生物技术有限公司 2022-02-11 CN disclosed
WO-2019141229-A1 COMPOUND AS PPAR AGONIST AND APPLICATION THEREOF 上海怡立舍生物技术有限公司 2019-07-25 WO disclosed
WO-2019141229-A1 COMPOUND AS PPAR AGONIST AND APPLICATION THEREOF 上海怡立舍生物技术有限公司 2019-07-25 WO disclosed
CN-108250058-A PPAR agonists and their use in the treatment of Alzheimer's disease and other diseases 上海怡立舍生物技术有限公司 2018-07-06 CN disclosed