SCHEMBL21187202

SCHEMBL21187202

COc1ccc(C2=CCC(NC(=O)OC(C)(C)C)CC2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.43
ALDH1A1 P00352 1/20 0.43
NAMPT P43490 1/20 0.42
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
DRD2 P14416 1/20 0.40
KDM1A O60341 1/20 0.40
MAOB P27338 1/20 0.40
EPHX2 P34913 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
EPHX1 P07099 1/20 0.40
PDE2A O00408 1/20 0.40
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
CKS1B P61024 1/20 0.39
SKP1 P63208 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL32677509 0.87 KDM4D (0.42) ALDH1A1NAMPTKMT2AL3MBTL1DRD2
SCHEMBL32677506 0.87 KDM4D (0.42) ALDH1A1NAMPTKMT2AL3MBTL1DRD2
SCHEMBL3701445 0.86 NAMPT (0.43) NAMPTKMT2AL3MBTL1DRD2KDM1A
SCHEMBL19380850 0.86 KMT2A (0.51) NAMPTKMT2AL3MBTL1DRD2KDM1A
SCHEMBL32677525 0.85 NAMPT (0.42) NAMPTKMT2AL3MBTL1DRD2KDM1A
SCHEMBL32677522 0.85 NAMPT (0.42) NAMPTKMT2AL3MBTL1DRD2KDM1A
SCHEMBL19380845 0.84 NAMPT (0.41) NAMPTKMT2AL3MBTL1DRD2KDM1A
SCHEMBL12321516 0.83 DRD2 (0.48) NAMPTKMT2AL3MBTL1DRD2KDM1A
SCHEMBL3707832 0.82 DRD2 (0.49) MAPTALDH1A1NAMPTKMT2AL3MBTL1
SCHEMBL32677535 0.81 NAMPT (0.38) NAMPTKMT2AL3MBTL1DRD2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111247119-B Amidine and guanidine derivatives, preparation method and application thereof in medicines 四川科伦博泰生物医药股份有限公司 2023-02-03 CN disclosed
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed