SCHEMBL21187253

SCHEMBL21187253

O=CC/C=C/c1csc2cc(Br)ccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.54
CA2 P00918 1/20 0.33
PRF1 P14222 1/20 0.32
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
ERN1 O75460 1/20 0.31
MAPT P10636 2/20 0.30
TP53 P04637 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPK1 P28482 1/20 0.30
KMT2A Q03164 1/20 0.30
TUBB4A P04350 1/20 0.30
TUBB P07437 1/20 0.30
TUBA3C P0DPH7 1/20 0.30
TUBA1B P68363 1/20 0.30
TUBA4A P68366 1/20 0.30
TUBB4B P68371 1/20 0.30
TUBB3 Q13509 1/20 0.30
TUBB2A Q13885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21177013 0.81 CYP2A6 (0.47) CYP2A6PRF1PTGS1PTGS2MAPT
SCHEMBL29452875 0.81 CYP2A6 (0.47) CYP2A6PRF1PTGS1PTGS2MAPT
SCHEMBL30197394 0.80 CYP2A6 (0.74) CYP2A6CA2PRF1ERN1ALDH1A1
SCHEMBL6811552 0.80 CYP2A6 (0.74) CYP2A6CA2PRF1ERN1ALDH1A1
SCHEMBL5539045 0.72 ERN1 (0.41) CYP2A6ERN1ALDH1A1
SCHEMBL5544825 0.72 HSP90AA1 (0.38) CYP2A6ERN1ALDH1A1MAPK1
SCHEMBL2022637 0.70 CYP2A6 (1.00) CYP2A6CA2PRF1ERN1MAPT
SCHEMBL6811378 0.70 CYP2A6 (0.50) CYP2A6CA2PTGS1PTGS2MAPT
SCHEMBL6811377 0.70 CYP2A6 (0.50) CYP2A6CA2PTGS1PTGS2MAPT
SCHEMBL2091129 0.69 GPR183 (0.39) CYP2A6ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141229-A1 COMPOUND AS PPAR AGONIST AND APPLICATION THEREOF 上海怡立舍生物技术有限公司 2019-07-25 WO disclosed