SCHEMBL6811552

SCHEMBL6811552

O=Cc1csc2cc(Br)ccc12

nearest known ligand 0.74

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.74
ERN1 O75460 5/20 0.44
PTPN1 P18031 1/20 0.39
PIM3 Q86V86 2/20 0.39
PIM1 P11309 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.35
CA2 P00918 1/20 0.35
ALDH1A1 P00352 1/20 0.34
MIF P14174 1/20 0.33
PRF1 P14222 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30197394 1.00 CYP2A6 (0.74) CYP2A6ERN1PTPN1PIM3PIM1
SCHEMBL2022637 0.85 CYP2A6 (1.00) CYP2A6ERN1PTPN1PIM3PIM1
SCHEMBL21187253 0.80 CYP2A6 (0.54) CYP2A6ERN1CA2ALDH1A1PRF1
SCHEMBL1121640 0.78 CYP2A6 (0.56) CYP2A6ERN1PTPN1CA2
SCHEMBL1121724 0.78 CYP2A6 (0.56) CYP2A6ERN1PTPN1CA2ALDH1A1
SCHEMBL6811378 0.77 CYP2A6 (0.50) CYP2A6CA2ALDH1A1
SCHEMBL6811377 0.77 CYP2A6 (0.50) CYP2A6CA2ALDH1A1
SCHEMBL25232594 0.76 CYP2A6 (0.46) CYP2A6CA2ALDH1A1MIF
SCHEMBL30445252 0.76 CYP2A6 (0.46) CYP2A6CA2ALDH1A1MIF
SCHEMBL17912642 0.74 CYP2A6 (0.61) CYP2A6ERN1PTPN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115626890-B Diamine monomer with bulky alkynyl side group, and preparation method and application thereof 波米科技有限公司 2023-05-16 CN claimed
CN-115626890-A Diamine monomer with bulky alkynyl side group and preparation method and application thereof 波米科技有限公司 2023-01-20 CN claimed
CN-115974762-B Diamine monomer with bulky alkynyl side group, polybenzoxazole precursor, photosensitive resin composition and application thereof 波米科技有限公司 2023-09-19 CN disclosed
CN-115626890-B Diamine monomer with bulky alkynyl side group, and preparation method and application thereof 波米科技有限公司 2023-05-16 CN disclosed
CN-115974762-A Diamine monomer with bulky alkynyl side group, polybenzoxazole precursor, photosensitive resin composition and application thereof 波米科技有限公司 2023-04-18 CN disclosed
CN-115626890-A Diamine monomer with bulky alkynyl side group and preparation method and application thereof 波米科技有限公司 2023-01-20 CN disclosed
CN-108250058-B PPAR agonists and their use in the treatment of Alzheimer's disease and other diseases 上海怡立舍生物技术有限公司 2022-02-11 CN disclosed
WO-2019141229-A1 COMPOUND AS PPAR AGONIST AND APPLICATION THEREOF 上海怡立舍生物技术有限公司 2019-07-25 WO disclosed
WO-2019141229-A1 COMPOUND AS PPAR AGONIST AND APPLICATION THEREOF 上海怡立舍生物技术有限公司 2019-07-25 WO disclosed
US-9993459-B2 Selective HDAC6 inhibitors and uses thereof UNIVERSITEIT GENT (BE) 2018-06-12 US disclosed
US-9993459-B2 Selective HDAC6 inhibitors and uses thereof UNIVERSITEIT GENT (BE) 2018-06-12 US disclosed
US-20170360748-A1 SELECTIVE HDAC6 INHIBITORS AND USES THEREOF UNIVERSITEIT GENT (BE) 2017-12-21 US disclosed
US-20170360748-A1 SELECTIVE HDAC6 INHIBITORS AND USES THEREOF UNIVERSITEIT GENT (BE) 2017-12-21 US disclosed
US-20170360748-A1 SELECTIVE HDAC6 INHIBITORS AND USES THEREOF UNIVERSITEIT GENT (BE) 2017-12-21 US disclosed
WO-2016110541-A1 SELECTIVE HDAC6 INHIBITORS AND USES THEREOF UNIVERSITEIT GENT (BE) 2016-07-14 WO disclosed
WO-2016110541-A1 SELECTIVE HDAC6 INHIBITORS AND USES THEREOF UNIVERSITEIT GENT (BE) 2016-07-14 WO disclosed
US-20040122001-A1 Pharmaceutical compounds ELI LILLY AND COMPANY 2004-06-24 US disclosed
EP-1345930-A2 PHARMACEUTICAL COMPOUNDS ELI LILLY AND COMPANY (US) 2003-09-24 EP disclosed
WO-2002050067-A2 PHARMACEUTICAL HETEROCYCLIC COMPOUNDS ELI LILLY AND COMPANY (US) 2002-06-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170360748-A1 SELECTIVE HDAC6 INHIBITORS AND USES THEREOF HDAC6, HDAC1, HDAC5 CYP2A6 4402/4885ERN1 2959/4885PTPN1 2399/4885
US-20040122001-A1 Pharmaceutical compounds CYP2D6, LPXN, CYP1B1 CYP2A6 39/4885ERN1 2132/4885PTPN1 1056/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.