SCHEMBL21187403

SCHEMBL21187403

c1nc(NC2CCCCC2)c2occc2n1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.69
HPGDS O60760 2/20 0.46
LMNA P02545 3/20 0.44
HTT P42858 3/20 0.44
HSD17B10 Q99714 2/20 0.44
PKM P14618 1/20 0.44
CD38 P28907 2/20 0.43
JAK2 O60674 2/20 0.43
JAK1 P23458 2/20 0.43
EGFR P00533 2/20 0.43
PAK1 Q13153 1/20 0.42
MEN1 O00255 1/20 0.41
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20273951 0.77 KMT2A (0.47) IRAK4HSD17B10JAK2KMT2A
SCHEMBL24023125 0.72 IRAK4 (0.42) IRAK4LMNAALDH1A1CYP3A4MAPK1
SCHEMBL20051446 0.72 IRAK4 (0.40) IRAK4ALDH1A1CYP3A4
SCHEMBL22872840 0.72 LMNA (0.55) IRAK4LMNAHSD17B10EGFRALDH1A1
SCHEMBL27504590 0.72 PDE5A (0.58) HPGDSHSD17B10CD38
SCHEMBL29118643 0.72 IRAK4 (0.49) IRAK4LMNAHTTEGFRALDH1A1
SCHEMBL30748895 0.72 IRAK4 (0.52) IRAK4LMNAHSD17B10EGFRUSP2
SCHEMBL3712626 0.72 IRAK4 (0.44) IRAK4HSD17B10JAK2KMT2A
SCHEMBL21318578 0.71 IRAK4 (0.77) IRAK4LMNAHSD17B10CD38MEN1
SCHEMBL22872893 0.70 MAP4K4 (0.49) HPGDSPKMJAK2JAK1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019143678-A1 DNA-PK INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2019-07-25 WO disclosed