SCHEMBL21230185

SCHEMBL21230185

CCCCN(CCC)C(=O)c1ccc(-c2noc(C(F)(F)F)c2C)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 3/20 0.35
HDAC1 Q13547 3/20 0.35
HDAC6 Q9UBN7 3/20 0.35
HDAC3 O15379 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
MLYCD O95822 1/20 0.34
ALDH1A1 P00352 3/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
KDM4E B2RXH2 1/20 0.34
TP53 P04637 2/20 0.34
RXFP1 Q9HBX9 2/20 0.34
POLB P06746 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21230173 0.94 ALDH1A1 (0.39) HDAC4HDAC1HDAC6HDAC3HDAC7
SCHEMBL21230117 0.87 ALDH1A1 (0.38) HDAC4HDAC1HDAC6HDAC3HDAC7
SCHEMBL19151672 0.86 ALDH1A1 (0.39) HDAC4HDAC1HDAC6HDAC3HDAC7
SCHEMBL8109881 0.85 HDAC4 (0.33) HDAC4HDAC1HDAC6HDAC3HDAC7
SCHEMBL3249605 0.81 ALDH1A1 (0.49) HDAC4HDAC1HDAC6HDAC3HDAC7
SCHEMBL3250456 0.78 HDAC6 (0.43) HDAC4HDAC1HDAC6HDAC3HDAC7
SCHEMBL3244594 0.78 ALDH1A1 (0.46) HDAC4HDAC1HDAC6HDAC3HDAC7
SCHEMBL3262869 0.77 HDAC4 (0.50) HDAC4HDAC1HDAC6HDAC3HDAC7
SCHEMBL18867357 0.77 NPC1 (0.47) HDAC4HDAC1HDAC6HDAC3HDAC7
SCHEMBL3247527 0.77 HDAC6 (0.42) HDAC4HDAC1HDAC6HDAC3HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3311813-B1 THERAPEUTIC ISOXAZOLE COMPOUNDS DART NEUROSCIENCE CAYMAN LTD (KY) 2019-08-07 EP disclosed