SCHEMBL21241228

SCHEMBL21241228

CNC(=N)Nc1ccc(C2=NNC(=O)CC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.51
PDE3B Q13370 11/20 0.51
LMNA P02545 2/20 0.47
MAPT P10636 2/20 0.47
NPY1R P25929 1/20 0.47
NPY2R P49146 1/20 0.47
PDE3A Q14432 10/20 0.46
PDE4A P27815 5/20 0.46
PDE4B Q07343 5/20 0.46
PDE4C Q08493 5/20 0.46
PDE4D Q08499 5/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
CYP2C19 P33261 1/20 0.46
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21241242 0.86 KCNH2 (0.52) KCNH2SMN1; SMN2PDE3BLMNAMAPT
SCHEMBL21241239 0.86 KCNH2 (0.52) KCNH2SMN1; SMN2PDE3BLMNAMAPT
SCHEMBL21241022 0.86 KCNH2 (0.52) KCNH2SMN1; SMN2PDE3BLMNAMAPT
SCHEMBL21241240 0.84 MAPT (0.51) KCNH2SMN1; SMN2PDE3BLMNAMAPT
SCHEMBL21241241 0.83 KCNH2 (0.58) KCNH2SMN1; SMN2PDE3BLMNAMAPT
SCHEMBL21241021 0.83 KCNH2 (0.52) KCNH2SMN1; SMN2PDE3BLMNAMAPT
SCHEMBL21241015 0.83 PDE3B (0.53) KCNH2SMN1; SMN2PDE3BLMNAMAPT
SCHEMBL6559298 0.82 KCNH2 (0.59) KCNH2SMN1; SMN2PDE3BLMNAMAPT
SCHEMBL22910067 0.81 KCNH2 (0.66) KCNH2SMN1; SMN2PDE3BLMNAMAPT
SCHEMBL10474308 0.80 KCNH2 (0.54) KCNH2SMN1; SMN2PDE3BLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3766872-A1 P2Y12 RECEPTOR ANTAGONIST CONTAINING GUANIDYL, AND PREPARATION METHOD AND USE THEREOF Anhui New Star Pharmaceutical Development Co., Ltd (CN) 2021-01-20 EP disclosed
WO-2019149259-A1 P2Y12 RECEPTOR ANTAGONIST CONTAINING GUANIDYL, AND PREPARATION METHOD AND USE THEREOF 安徽省新星药物开发有限责任公司 2019-08-08 WO disclosed