SCHEMBL21243055

SCHEMBL21243055

CCON(C)C(=O)c1cccc2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC25B P30305 2/20 0.54
NR4A1 P22736 1/20 0.49
NR4A2 P43354 1/20 0.49
NR4A3 Q92570 1/20 0.49
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
PTPN1 P18031 1/20 0.47
PLK1 P53350 1/20 0.47
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
CDC25A P30304 1/20 0.47
CDC25C P30307 1/20 0.47
CNR1 P21554 2/20 0.46
CNR2 P34972 2/20 0.46
TSHR P16473 2/20 0.46
GMNN O75496 2/20 0.45
LMNA P02545 2/20 0.45
POLB P06746 2/20 0.45
MAPT P10636 2/20 0.45
HPGD P15428 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14588679 0.89 CNR2 (0.52) CDC25BNR4A1NR4A2NR4A3MEN1
SCHEMBL1515779 0.83 NR4A1 (0.52) CDC25BNR4A1NR4A2NR4A3MEN1
SCHEMBL14620600 0.82 CDC25B (0.46) CDC25BNR4A1NR4A2NR4A3MEN1
SCHEMBL27794823 0.81 CDC25B (0.50) CDC25BNR4A1NR4A2NR4A3MEN1
SCHEMBL18652132 0.80 NR4A1 (0.52) CDC25BNR4A1NR4A2NR4A3MEN1
SCHEMBL10407111 0.79 NR4A1 (0.59) CDC25BNR4A1NR4A2NR4A3MEN1
SCHEMBL3624003 0.78 OPRM1 (0.56) CDC25BNR4A1NR4A2NR4A3MEN1
Hydrochloric Acid SCHEMBL11683665 0.77 NR4A1 (0.56) CDC25BNR4A1NR4A2NR4A3MEN1
SCHEMBL12984879 0.77 SMPD2 (0.44) CDC25BNR4A1NR4A2NR4A3MEN1
SCHEMBL28713330 0.76 CDC25B (0.49) CDC25BNR4A1NR4A2NR4A3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3842424-A1 MAP KINASE MODULATORS AND USES THEREOF IN THE TRETAMENT OF TAUOPATHIES The Trustees of Columbia University in the City of New York (US) 2021-06-30 EP disclosed
EP-3521284-A1 PYRAZINE COMPOUNDS AS MAP KINASE MODULATORS AND USES THEREOF The Trustees of Columbia University in the City of New York (US) 2019-08-07 EP disclosed