SCHEMBL21246631

SCHEMBL21246631

COc1cc(NSc2ccc(C)cc2)cc(C(=O)NCc2cccnc2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.58
MMP13 P45452 1/20 0.58
SMN1; SMN2 Q16637 3/20 0.56
LMNA P02545 2/20 0.56
GLA P06280 1/20 0.56
POLB P06746 1/20 0.56
HPGD P15428 1/20 0.56
CYP1A2 P05177 3/20 0.53
CYP3A4 P08684 3/20 0.53
TSHR P16473 2/20 0.53
BLM P54132 1/20 0.53
ALDH1A1 P00352 3/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
USP2 O75604 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
CYP2C19 P33261 2/20 0.52
KCNJ1 P48048 1/20 0.49
CYP2C9 P11712 1/20 0.49
RECQL P46063 1/20 0.48
MAPK1 P28482 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21246550 0.89 LMNA (0.61) MMP13SMN1; SMN2LMNAGLAPOLB
SCHEMBL21246549 0.87 LMNA (0.58) MMP13SMN1; SMN2LMNAGLAPOLB
SCHEMBL21246551 0.87 HPGD (0.58) MMP13SMN1; SMN2LMNAGLAPOLB
SCHEMBL21246540 0.85 LMNA (0.61) MMP13SMN1; SMN2LMNAGLAPOLB
SCHEMBL29437179 0.82 NAMPT (0.69) GAAMMP13ALDH1A1KCNJ1HTT
SCHEMBL22729253 0.82 NAMPT (0.69) GAAMMP13ALDH1A1KCNJ1HTT
SCHEMBL21246545 0.81 CYP1A2 (0.67) GAAMMP13SMN1; SMN2LMNAGLA
SCHEMBL21246582 0.79 GAA (0.67) GAAMMP13SMN1; SMN2LMNAGLA
SCHEMBL21246578 0.79 LMNA (0.55) MMP13SMN1; SMN2LMNAGLAPOLB
SCHEMBL21246562 0.79 LMNA (0.63) GAAMMP13SMN1; SMN2LMNAGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3747866-A1 BENZAMIDE COMPOUND AND PREPARATION METHOD, USE, AND PHARMACEUTICAL COMPOSITION THEREOF INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2020-12-09 EP disclosed
WO-2019149223-A1 BENZAMIDE COMPOUND AND PREPARATION METHOD, USE, AND PHARMACEUTICAL COMPOSITION THEREOF 中国医学科学院药物研究所 2019-08-08 WO disclosed