SCHEMBL21248036

SCHEMBL21248036

Cc1ccc(NC(=O)c2ccc(CBr)cc2)cc1Nc1nccc(-c2cccnc2)n1

nearest known ligand 0.84

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 15/20 0.84
ABL1 P00519 11/20 0.84
KIT P10721 9/20 0.84
BCR P11274 8/20 0.82
PDGFRB P09619 5/20 0.82
EGFR P00533 2/20 0.80
PRKCA P17252 1/20 0.80
KDR P35968 2/20 0.75
PLK4 O00444 1/20 0.74
DDX3X O00571 1/20 0.74
GAK O14976 1/20 0.74
SLC22A2 O15244 1/20 0.74
MAPK13 O15264 1/20 0.74
CA12 O43570 1/20 0.74
SLC22A3 O75751 1/20 0.74
ABCB11 O95342 1/20 0.74
CA1 P00915 1/20 0.74
CA2 P00918 1/20 0.74
LMNA P02545 1/20 0.74
ALB P02768 1/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27962634 0.93 PDGFRA (0.81) PDGFRAABL1KITBCRPDGFRB
SCHEMBL805395 0.92 PDGFRA (0.85) PDGFRAABL1KITBCRPDGFRB
SCHEMBL27804782 0.92 PDGFRA (0.85) PDGFRAABL1KITBCRPDGFRB
SCHEMBL25281830 0.91 PDGFRA (1.00) PDGFRAABL1KITBCRPDGFRB
SCHEMBL14292529 0.91 PDGFRA (0.84) PDGFRAABL1KITBCRPDGFRB
SCHEMBL723757 0.91 PDGFRA (1.00) PDGFRAABL1KITBCRPDGFRB
SCHEMBL29628979 0.91 PDGFRA (1.00) PDGFRAABL1KITBCRPDGFRB
Hydrochloric Acid SCHEMBL4396677 0.90 PDGFRA (0.98) PDGFRAABL1KITBCRPDGFRB
SCHEMBL3065290 0.90 PDGFRA (0.89) PDGFRAABL1KITBCRPDGFRB
SCHEMBL9820 0.90 PDGFRA (1.00) PDGFRAABL1KITBCRPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240257921-A1 COMPUTATIONAL GENERATION OF CHEMICAL SYNTHESIS ROUTES AND METHODS STANFORD RES INST INT (US) 2024-08-01 US disclosed
US-11961595-B2 Computational generation of chemical synthesis routes and methods SRI INTERNATIONAL (US) 2024-04-16 US disclosed
US-20210065851-A1 COMPUTATIONAL GENERATION OF CHEMICAL SYNTHESIS ROUTES AND METHODS SRI INTERNATIONAL 2021-03-04 US disclosed
CN-112272764-A Computational generation of chemical synthetic routes and methods 斯坦福国际研究院 2021-01-26 CN disclosed
EP-3746772-A1 COMPUTATIONAL GENERATION OF CHEMICAL SYNTHESIS ROUTES AND METHODS Madrid, Peter (US) 2020-12-09 EP disclosed
WO-2019156872-A9 COMPUTATIONAL GENERATION OF CHEMICAL SYNTHESIS ROUTES AND METHODS MADRID PETER (US) 2019-10-03 WO disclosed
WO-2019156872-A1 COMPUTATIONAL GENERATION OF CHEMICAL SYNTHESIS ROUTES AND METHODS MADRID PETER (US) 2019-08-15 WO disclosed