SCHEMBL21274152

SCHEMBL21274152

NC(=O)OCC1CCC(=O)N1

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 18/20 0.42
IRAK1 P51617 1/20 0.40
MGLL Q99685 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23725735 1.00 IRAK4 (0.42) IRAK4IRAK1MGLL
SCHEMBL9994585 0.85 MGLL (0.41) IRAK4IRAK1MGLL
SCHEMBL9994588 0.84 MGLL (0.40) IRAK4IRAK1MGLL
SCHEMBL18009354 0.81 MGLL (0.39) IRAK4IRAK1MGLL
SCHEMBL1715768 0.79
SCHEMBL19973031 0.79
SCHEMBL18014839 0.76 HCAR2 (0.40) IRAK4IRAK1MGLL
SCHEMBL18009241 0.74 HCAR2 (0.38) IRAK4IRAK1MGLL
SCHEMBL18009250 0.74 HCAR2 (0.38) IRAK4IRAK1MGLL
SCHEMBL18009233 0.74 HCAR2 (0.38) IRAK4IRAK1MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118084940-A PD-1/PD-L1 inhibitors 吉利德科学公司 2024-05-28 CN disclosed
CN-117412959-A Substituted 1-aryl-1 '-heteroaryl compounds, substituted 1,1' -biaryl compounds, and methods of use thereof 爱彼特生物制药公司 2024-01-16 CN disclosed
CN-112041311-B PD-1/PD-L1 inhibitors 吉利德科学公司 2023-10-03 CN disclosed
EP-4227302-A1 PD-1/PD-L1 INHIBITORS Gilead Sciences, Inc. (US) 2023-08-16 EP disclosed
US-20230212155-A1 PD-1/PD-L1 INHIBITORS GILEAD SCIENCES, INC. 2023-07-06 US disclosed
EP-4169925-A2 PROCESS TO MAKE N-SUBSTITUTED TETRAHYDROTHIENOPYRIDINE DERIVATIVES Novartis AG (CH) 2023-04-26 EP disclosed
EP-3752501-B1 PD-1/PD-L1 INHIBITORS GILEAD SCIENCES INC (US) 2023-04-19 EP disclosed
US-11555029-B2 PD-1/PD-L1 inhibitors GILEAD SCIENCES, INC. (US) 2023-01-17 US disclosed
CN-115413275-A Substituted 1,1 , -biphenyl compounds and methods of use thereof 爱彼特生物制药公司 2022-11-29 CN disclosed
US-20210053946-A1 PD-1/PD-L1 INHIBITORS GILEAD SCIENCES, INC. (US) 2021-02-25 US disclosed
EP-3752501-A1 PD-1/PD-L1 INHIBITORS GILEAD SCIENCES, INC. (US) 2020-12-23 EP disclosed
CN-112041311-A PD-1/PD-L1 inhibitors 吉利德科学公司 2020-12-04 CN disclosed
CN-111712494-A PD-1/PD-L1 inhibitors 吉利德科学公司 2020-09-25 CN disclosed
US-10710986-B2 PD-1/PD-L1 inhibitors GILEAD SCIENCES, INC. (US) 2020-07-14 US disclosed
US-20190270727-A1 PD-1/PD-L1 INHIBITORS GILEAD SCIENCES, INC. 2019-09-05 US disclosed
WO-2019160882-A1 PD-1/PD-L1 INHIBITORS GILEAD SCIENCES, INC. (US) 2019-08-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11555029-B2 PD-1/PD-L1 inhibitors PDCD1, CD274, PDCD1LG2 IRAK4 1881/4885IRAK1 1253/4885MGLL 1243/4885
US-20230212155-A1 PD-1/PD-L1 INHIBITORS PDCD1, CD274, PDCD1LG2 IRAK4 1881/4885IRAK1 1253/4885MGLL 1243/4885
US-20210053946-A1 PD-1/PD-L1 INHIBITORS PDCD1, CD274, PDCD1LG2 IRAK4 1881/4885IRAK1 1253/4885MGLL 1243/4885
US-10710986-B2 PD-1/PD-L1 inhibitors PDCD1, CD274, PDCD1LG2 IRAK4 1881/4885IRAK1 1253/4885MGLL 1243/4885
US-20190270727-A1 PD-1/PD-L1 INHIBITORS PDCD1, CD274, PDCD1LG2 IRAK4 1881/4885IRAK1 1253/4885MGLL 1243/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.