SCHEMBL21275464

SCHEMBL21275464

Nc1ccc(N2CCC(O)CC2I)cn1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 6/20 0.44
CHRNA4 P43681 6/20 0.44
ALOX5AP P20292 1/20 0.35
FEN1 P39748 1/20 0.35
PIK3CA P42336 1/20 0.34
MTOR P42345 1/20 0.34
CHRNB4 P30926 4/20 0.34
CHRNA3 P32297 4/20 0.34
PIK3CD O00329 1/20 0.33
KDM4E B2RXH2 1/20 0.32
GCKR Q14397 5/20 0.31
GCK P35557 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23104482 0.83 CHRNB2 (0.44) CHRNB2CHRNA4ALOX5APFEN1PIK3CA
SCHEMBL23089144 0.83 CHRNB2 (0.44) CHRNB2CHRNA4ALOX5APFEN1PIK3CA
SCHEMBL29814518 0.83 CHRNB2 (0.44) CHRNB2CHRNA4ALOX5APFEN1PIK3CA
SCHEMBL619825 0.75 MAPT (0.49) CHRNB2CHRNA4ALOX5APFEN1PIK3CA
SCHEMBL29891246 0.75 MAPT (0.49) CHRNB2CHRNA4ALOX5APFEN1PIK3CA
SCHEMBL13769145 0.74 CDK1 (0.49) CHRNB2CHRNA4ALOX5APFEN1PIK3CA
SCHEMBL4528273 0.74 CDK1 (0.49) CHRNB2CHRNA4ALOX5APFEN1PIK3CA
SCHEMBL29618159 0.74 CDK1 (0.49) CHRNB2CHRNA4ALOX5APFEN1PIK3CA
SCHEMBL4721289 0.74 CDK1 (0.49) CHRNB2CHRNA4ALOX5APFEN1PIK3CA
SCHEMBL23089266 0.71 MAPT (0.45) CHRNB2CHRNA4ALOX5APFEN1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752491-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS Nuvation Bio Inc. (US) 2020-12-23 EP disclosed
WO-2019161224-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS GiraFpharma LLC (US) 2019-08-22 WO disclosed