SCHEMBL21278024

SCHEMBL21278024

Cc1cccc(-c2nc3n(c2-c2ccnc(-c4ccc([S+](C)[O-])cc4)c2)C2CCC3C2)n1

nearest known ligand 0.75

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 20/20 0.75
KDR P35968 9/20 0.75
MAPK14 Q16539 5/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20074514 1.00 TGFBR1 (0.75) TGFBR1KDRMAPK14
SCHEMBL21277863 1.00 TGFBR1 (0.75) TGFBR1KDRMAPK14
SCHEMBL21278023 0.92 TGFBR1 (0.76) TGFBR1KDRMAPK14
SCHEMBL20074460 0.89 TGFBR1 (0.80) TGFBR1KDRMAPK14
SCHEMBL20074464 0.86 TGFBR1 (1.00) TGFBR1KDRMAPK14
SCHEMBL20074459 0.86 TGFBR1 (1.00) TGFBR1KDRMAPK14
SCHEMBL20074503 0.86 TGFBR1 (1.00) TGFBR1KDRMAPK14
SCHEMBL20074582 0.85 TGFBR1 (1.00) TGFBR1KDRMAPK14
SCHEMBL20074718 0.85 TGFBR1 (1.00) TGFBR1KDRMAPK14
SCHEMBL20074722 0.85 TGFBR1 (1.00) TGFBR1KDRMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3527570-A1 FIVE-MEMBERED HETEROARYL RING BRIDGED RING DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF Jiangsu Hengrui Medicine Co., Ltd. (CN) 2019-08-21 EP disclosed