SCHEMBL21290150

SCHEMBL21290150

COc1cc(-c2cc3ccccc3cn2)ccc1-c1ccccc1Br

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.56
RAB9A P51151 7/20 0.56
CASP3 P42574 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
S1PR1 P21453 1/20 0.42
IDO1 P14902 5/20 0.41
TDO2 P48775 5/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
RAC1 P63000 2/20 0.40
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
ALOX5AP P20292 1/20 0.39
FEN1 P39748 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21290361 0.82 POLB (0.43) NPC1RAB9AS1PR1KDM4EALDH1A1
SCHEMBL27993895 0.81 NPC1 (0.69) NPC1RAB9ACASP3SENP7S1PR1
SCHEMBL21290393 0.80 ERN1 (0.46) NPC1RAB9AKDM4EALDH1A1SMN1; SMN2
SCHEMBL23956222 0.80 NPC1 (0.67) NPC1RAB9AKDM4EALDH1A1SMN1; SMN2
SCHEMBL21290358 0.80 PDE4D (0.42) NPC1RAB9AS1PR1KDM4EALDH1A1
SCHEMBL21290156 0.79 NPC1 (0.39) NPC1RAB9AIDO1TDO2KDM4E
SCHEMBL23956198 0.78 ALOX5AP (0.37) NPC1RAB9AS1PR1TDO2KDM4E
SCHEMBL21289974 0.78 ACACA (0.48) KDM4EALDH1A1SMN1; SMN2RAC1TP53
SCHEMBL23956286 0.77 NPC1 (0.50) NPC1RAB9ACASP3SENP7IDO1
SCHEMBL21290149 0.77 IDO1 (0.48) NPC1RAB9AIDO1TDO2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
EP-3601304-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2021-10-27 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed