SCHEMBL21290780

SCHEMBL21290780

CCNCCc1cnn[nH]1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 5/20 0.41
HRH3 Q9Y5N1 5/20 0.41
HTR2A P28223 2/20 0.33
CCNK O75909 1/20 0.33
CDK12 Q9NYV4 1/20 0.33
HTT P42858 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
MPO P05164 1/20 0.30
GLA P06280 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21322194 0.87 HRH4 (0.42) HRH4HRH3MEN1KMT2AALDH1A1
SCHEMBL2580256 0.81
SCHEMBL21290462 0.80 HRH4 (0.45) HRH4HRH3ALDH1A1CYP2C19
SCHEMBL23948654 0.80
SCHEMBL16629040 0.76
SCHEMBL1998113 0.76 ADH1B (0.31)
SCHEMBL21573784 0.73 HRH4 (0.39) HRH4HRH3MEN1KMT2AALDH1A1
SCHEMBL19764586 0.73 HRH4 (0.51) HRH4HRH3
SCHEMBL1232300 0.72 HRH3 (0.42) HRH4HRH3KMT2A
SCHEMBL2576444 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019204609-A1 PD-1/PD-L1 INHIBITORS GILEAD SCIENCES, INC. (US) 2019-10-24 WO disclosed
WO-2019160882-A1 PD-1/PD-L1 INHIBITORS GILEAD SCIENCES, INC. (US) 2019-08-22 WO disclosed