SCHEMBL2129641

SCHEMBL2129641

CCCc1nc2c(C)cc(C(=O)O)cc2n1Cc1ccc(-c2ccccc2C#N)cc1

nearest known ligand 0.65

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 18/20 0.65
AGTR2 P50052 5/20 0.63
PPARG P37231 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14775798 0.91 AGTR1 (0.60) AGTR1AGTR2PPARG
SCHEMBL8266757 0.87 AGTR1 (0.82) AGTR1AGTR2PPARG
SCHEMBL29387259 0.87 AGTR1 (0.82) AGTR1AGTR2PPARG
SCHEMBL3686030 0.86 AGTR1 (0.62) AGTR1AGTR2
SCHEMBL8003999 0.86 PPARG (0.72) AGTR1AGTR2PPARG
SCHEMBL3681150 0.85 AGTR1 (0.53) AGTR1AGTR2PPARG
SCHEMBL8096420 0.85 PPARG (0.63) AGTR1AGTR2PPARG
SCHEMBL8942730 0.83 PPARG (0.61) AGTR1AGTR2PPARG
SCHEMBL12606480 0.83 AGTR1 (0.73) AGTR1AGTR2
SCHEMBL3638002 0.83 AGTR1 (0.64) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2443094-B1 PROCESS FOR THE PREPARATION OF TELMISARTAN KRKA TOVARNA ZDRAVIL D D NOVO MESTO (SI) 2013-03-20 EP disclosed
EP-2443094-A2 PROCESS FOR THE PREPARATION OF TELMISARTAN Krka Tovarna Zdravil, D.D., Novo Mesto (SI) 2012-04-25 EP disclosed
WO-2010146187-A2 PROCESS FOR THE PREPARATION OF TELMISARTAN KRKA, TOVARNA ZDRAVIL, D.D., NOVO MESTO (SI) 2010-12-23 WO disclosed
WO-2009116089-A2 NOVEL INTERMEDIATES AND METHOD FOR SYNTHESIS OF 4'-[(1,4'-DIMETHYL-2'-PROPYL-[2,6'- BI-1HBENZIMIDAZOL]-L-YL)METHYL]-1,1-BIPHENYL]-2-CARBOXYLIC ACID. IPCA LABORATORIES LIMITED (IN) 2009-09-24 WO disclosed