SCHEMBL21323318

SCHEMBL21323318

O=C(/C=C/c1cc(Cl)cc(Cl)c1)N1CCC2CN(C(=O)c3ccc4[nH]nnc4c3)C[C@H]2CC1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 5/20 0.54
ATXN2 Q99700 2/20 0.54
GPR183 P32249 8/20 0.40
CNR2 P34972 2/20 0.40
KCNH2 Q12809 2/20 0.40
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16962846 1.00 ENPP2 (0.54) ENPP2ATXN2GPR183CNR2KCNH2
SCHEMBL16962843 1.00 ENPP2 (0.54) ENPP2ATXN2GPR183CNR2KCNH2
SCHEMBL16961555 0.97 ENPP2 (0.51) ENPP2ATXN2GPR183CNR2KCNH2
SCHEMBL16961558 0.97 ENPP2 (0.51) ENPP2ATXN2GPR183CNR2KCNH2
SCHEMBL16961552 0.97 ENPP2 (0.51) ENPP2ATXN2GPR183CNR2KCNH2
SCHEMBL16961561 0.97 ENPP2 (0.51) ENPP2ATXN2GPR183CNR2KCNH2
SCHEMBL17310920 0.95 ENPP2 (0.51) ENPP2ATXN2GPR183CNR2KCNH2
SCHEMBL16962435 0.95 ENPP2 (0.51) ENPP2ATXN2GPR183CNR2KCNH2
SCHEMBL17310921 0.95 ENPP2 (0.51) ENPP2ATXN2GPR183CNR2KCNH2
SCHEMBL17310922 0.95 ENPP2 (0.51) ENPP2ATXN2GPR183CNR2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900669-B1 HEXAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AND RELATED COMPOUNDS AS AUTOTAXIN (ATX) INHIBITORS AND AS INHIBITORS OF THE LYSOPHOSPHATIDIC ACID (LPA) PRODUCTION FOR TREATING E.G. RENAL DISEASES HOFFMANN LA ROCHE (CH) 2019-09-04 EP disclosed