SCHEMBL21349331

SCHEMBL21349331

C=CCn1c(=O)c2cnc(SC)nc2n1-c1ccc2c(n1)C(CC)CC2

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
WEE1 P30291 20/20 0.52
PLK1 P53350 2/20 0.43
EGFR P00533 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAP3K19 Q56UN5 1/20 0.42
PLK3 Q9H4B4 1/20 0.42
PLK2 Q9NYY3 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21349629 0.89 WEE1 (0.64) WEE1PLK1EGFRCYP3A4MAP3K19
SCHEMBL25828125 0.89 WEE1 (0.43) WEE1PLK1
SCHEMBL22851870 0.85 WEE1 (0.58) WEE1PLK1EGFRCYP3A4MAP3K19
SCHEMBL21350111 0.79 WEE1 (0.64) WEE1PLK1EGFRCYP3A4MAP3K19
SCHEMBL25576991 0.79 WEE1 (0.64) WEE1PLK1EGFRCYP3A4MAP3K19
SCHEMBL21333353 0.79 WEE1 (0.65) WEE1PLK1EGFRCYP3A4MAP3K19
SCHEMBL24881605 0.79 WEE1 (0.65) WEE1PLK1EGFRCYP3A4MAP3K19
SCHEMBL21349330 0.79 WEE1 (0.65) WEE1PLK1EGFRCYP3A4MAP3K19
SCHEMBL21350035 0.79 WEE1 (0.65) WEE1PLK1EGFRCYP3A4MAP3K19
SCHEMBL30984877 0.79 WEE1 (0.65) WEE1PLK1EGFRCYP3A4MAP3K19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023016417-A1 1,2-DIHYDRO-3H-PYRAZOL[3,4-D]PYRIMIDIN-3-ONE COMPOUND AS WEE-1 INHIBITOR 微境生物医药科技(上海)有限公司 2023-02-16 WO disclosed
WO-2023280180-A1 FUSED RING COMPOUND AS WEE-1 INHIBITOR 微境生物医药科技(上海)有限公司 2023-01-12 WO disclosed
WO-2021252667-A1 METHODS OF MAKING WEE1 INHIBITOR COMPOUNDS RECURIUM IP HOLDINGS, LLC (US) 2021-12-16 WO disclosed
WO-2019173082-A1 SUBSTITUTED L,2-DIHYDRO-3H-PYRAZOLO[3,4-D]PYRIMIDIN-3-ONES Zeno Royalties & Milestones, LLC (US) 2019-09-12 WO disclosed