SCHEMBL21358271

SCHEMBL21358271

Nc1ncc(N2CCOCC2)c(N)n1

nearest known ligand 0.74

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHFR P00374 16/20 0.74
PIK3CA P42336 4/20 0.56
MTOR P42345 3/20 0.52
PIK3R1 P27986 2/20 0.52
RICTOR Q6R327 1/20 0.50
RPTOR Q8N122 1/20 0.50
MAPKAP1 Q9BPZ7 1/20 0.50
MLST8 Q9BVC4 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1776787 0.83 DHFR (0.65) DHFR
SCHEMBL4610473 0.82 DHFR (0.61) DHFRPIK3CAMTORPIK3R1RICTOR
Water SCHEMBL28223989 0.81 DHFR (0.63) DHFR
SCHEMBL7165357 0.81 DHFR (0.63) DHFR
SCHEMBL31649797 0.79 DHFR (0.51) DHFRPIK3CAMTORPIK3R1
SCHEMBL9167447 0.79 DHFR (0.59) DHFR
SCHEMBL28324074 0.79 DHFR (0.65) DHFR
SCHEMBL20734783 0.78 DHFR (1.00) DHFR
SCHEMBL2558872 0.78 DHFR (0.60) DHFRPIK3CAMTORPIK3R1RICTOR
SCHEMBL855868 0.77 PIK3CA (0.68) DHFRPIK3CAMTORPIK3R1RICTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019177375-A1 2, 4, 5-SUBSTITUTED PYRIMIDINE DERIVATIVES, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING CANCER COMPRISING SAME AS ACTIVE INGREDIENT 포로노이바이오 주식회사 2019-09-19 WO disclosed