SCHEMBL21359992

SCHEMBL21359992

C=CCC1CCN(C(=O)O)C1(C)C(=O)OC

nearest known ligand 0.32

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.31
CTSG P08311 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP3A4 P08684 1/20 0.31
MAPT P10636 1/20 0.31
TSHR P16473 1/20 0.31
KMT2A Q03164 1/20 0.31
FAAH O00519 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21367010 0.83 EPHX1 (0.33) ELANECTSGKDM4EALDH1A1CYP3A4
SCHEMBL21358152 0.81
SCHEMBL21359989 0.79
SCHEMBL21360032 0.72 ELANE (0.41) ELANECTSGFAAH
SCHEMBL15483731 0.70 KMT2A (0.32) KDM4EMEN1ALDH1A1CYP3A4MAPT
SCHEMBL21366841 0.69 ELANE (0.30) ELANECTSG
SCHEMBL22968579 0.68 GAA (0.32)
SCHEMBL22968577 0.68 GAA (0.32)
SCHEMBL21366843 0.67 GAA (0.31)
SCHEMBL21244731 0.65 FAAH (0.30) FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3765006-A1 ARGINASE INHIBITORS AND METHODS OF USE Merck Sharp&Dohme Corp. (US) 2021-01-20 EP disclosed
WO-2019177873-A1 ARGINASE INHIBITORS AND METHODS OF USE MERCK SHARP & DOHME CORP. (US) 2019-09-19 WO disclosed