SCHEMBL21362614

SCHEMBL21362614

O=C(c1ccc(Cl)cc1)c1cc(Cl)ccc1Br

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.52
KCNH2 Q12809 10/20 0.52
SRD5A2 P31213 2/20 0.50
NR4A1 P22736 1/20 0.50
KMT2A Q03164 2/20 0.49
MAPK1 P28482 1/20 0.48
RAB9A P51151 2/20 0.46
MAPT P10636 1/20 0.46
MEN1 O00255 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2875670 0.89 TP53 (0.65) TP53KCNH2NR4A1KMT2AMAPT
SCHEMBL20158110 0.86 MDM2 (0.46) TP53KCNH2SRD5A2NR4A1KMT2A
SCHEMBL28039223 0.85 MAPT (0.68) KCNH2KMT2AMAPK1RAB9AMAPT
SCHEMBL10599055 0.85 SRD5A2 (0.54) TP53SRD5A2NR4A1KMT2AMAPK1
SCHEMBL9280669 0.82 POLB (0.71) KCNH2KMT2AMAPK1RAB9AMAPT
SCHEMBL9281265 0.81 NR4A1 (0.65) TP53SRD5A2NR4A1KMT2AMAPK1
SCHEMBL29928911 0.81 NR4A1 (0.65) TP53SRD5A2NR4A1KMT2AMAPK1
SCHEMBL7466437 0.80 ALDH1A1 (0.61) TP53SRD5A2NR4A1KMT2AMAPK1
SCHEMBL9779330 0.78 CA1 (0.62) TP53KCNH2SRD5A2NR4A1KMT2A
SCHEMBL5022620 0.78 ALDH1A1 (0.53) TP53SRD5A2MAPK1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed