SCHEMBL21362691

SCHEMBL21362691

CCSCc1ccc(C(=O)c2ccc(F)cc2F)c(-c2cn(C)c(=O)cc2CNC(=O)OC(C)(C)C)c1

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 7/20 0.38
BRD4 O60885 11/20 0.35
GRM2 Q14416 1/20 0.33
PDE10A Q9Y233 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21564880 0.92 BRD4 (0.32) MAPK14BRD4GRM2
SCHEMBL21564931 0.92 P2RX7 (0.34) MAPK14BRD4GRM2
SCHEMBL21564927 0.88 IDO1 (0.34) BRD4GRM2
SCHEMBL21362077 0.88 BRD4 (0.40) MAPK14BRD4GRM2
SCHEMBL21564746 0.87 IDO1 (0.37)
SCHEMBL21564908 0.87 IDO1 (0.39)
SCHEMBL21564922 0.87 POLB (0.37)
SCHEMBL21564753 0.85 POLB (0.38)
SCHEMBL21564907 0.84 P2RX7 (0.36) BRD4GRM2
SCHEMBL20157909 0.81 BRD4 (0.34) MAPK14BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed