SCHEMBL21370838

SCHEMBL21370838

O=C1/C=C/C=C\C[C@H](O)CCOC(=O)c2c(O)cc(O)c(Cl)c2C1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 4/20 0.51
HSP90AA1 P07900 2/20 0.51
MAPT P10636 2/20 0.51
ACLY P53396 2/20 0.51
GAA P10253 1/20 0.51
RAB9A P51151 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
NLRP3 Q96P20 1/20 0.51
CBR1 P16152 1/20 0.51
PTGS2 P35354 1/20 0.51
FTO Q9C0B1 1/20 0.51
MEN1 O00255 1/20 0.51
ALDH1A1 P00352 1/20 0.51
HPGD P15428 1/20 0.51
KMT2A Q03164 1/20 0.51
STAT6 P42226 7/20 0.35
SMAD3 P84022 7/20 0.35
SMAD2 Q15796 7/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18966859 0.81 HSP90AB1 (0.50) HSP90AB1HSP90AA1MAPTACLYGAA
SCHEMBL10098854 0.80 HSP90AB1 (0.70) HSP90AB1HSP90AA1MAPTACLYGAA
SCHEMBL2622305 0.78 HSP90AB1 (0.76) HSP90AB1HSP90AA1MAPTACLYGAA
SCHEMBL19418358 0.77 HSP90AB1 (0.71) HSP90AB1HSP90AA1MAPTACLYGAA
SCHEMBL10150174 0.76 HSP90AB1 (0.66) HSP90AB1HSP90AA1MAPTACLYGAA
SCHEMBL19418377 0.75 HSP90AB1 (0.55) HSP90AB1HSP90AA1MAPTACLYGAA
SCHEMBL13748257 0.73 HSP90AB1 (0.66) HSP90AB1HSP90AA1MAPTACLYGAA
SCHEMBL14212853 0.73 HSP90AB1 (0.66) HSP90AB1HSP90AA1MAPTACLYGAA
SCHEMBL10293251 0.71 HSP90AB1 (0.70) HSP90AB1HSP90AA1MAPTACLYGAA
SCHEMBL19418322 0.71 HSP90AB1 (0.70) HSP90AB1HSP90AA1MAPTACLYGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020110056-A1 COMPOUNDS USEFUL IN HIV THERAPY GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2020-06-04 WO disclosed
EP-3181564-B1 AMINOPYRIMIDINE COMPOUNDS AS INHIBITORS OF T790M CONTAINING EGFR MUTANTS HOFFMANN LA ROCHE (CH) 2019-09-18 EP disclosed