SCHEMBL21372258

SCHEMBL21372258

CSC1CN(C(=O)C2CC2)C1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 10/20 0.50
CHRNA3 P32297 10/20 0.50
CHRNA4 P43681 10/20 0.50
CHRNB3 Q05901 5/20 0.50
CHRNA6 Q15825 5/20 0.50
CHRNB4 P30926 5/20 0.48
CHRNA7 P36544 5/20 0.48
HSD11B1 P28845 5/20 0.45
HPGD P15428 1/20 0.45
MAPT P10636 1/20 0.43
HSD11B2 P80365 2/20 0.42
HRH3 Q9Y5N1 1/20 0.40
HTT P42858 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24456544 0.76 RECQL (0.40) ALDH1A1TSHR
SCHEMBL16829688 0.75
SCHEMBL19014334 0.75
SCHEMBL10140410 0.75 CHRNB2 (0.56) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6
SCHEMBL24706079 0.72 CHRNB2 (0.58) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6
SCHEMBL26691462 0.71 CHRNB2 (0.52) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6
SCHEMBL15161321 0.70 CHRNB2 (0.56) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6
SCHEMBL3283590 0.70 HPGD (0.56) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6
SCHEMBL21891883 0.70 CHRNB2 (0.50) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6
SCHEMBL17816044 0.70 CHRNB2 (0.50) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3180344-B1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES USEFUL FOR INHIBITING JANUS KINASE PFIZER (US) 2019-09-18 EP disclosed