SCHEMBL21373095

SCHEMBL21373095

ONC(=Nc1ccc(Cl)c(Cl)c1)c1ccnc2nc[nH]c12

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 9/20 0.39
TDO2 P48775 2/20 0.37
HTR3E A5X5Y0 2/20 0.36
HTR3B O95264 2/20 0.36
HTR3A P46098 2/20 0.36
HTR3D Q70Z44 2/20 0.36
HTR3C Q8WXA8 2/20 0.36
POLA1 P09884 2/20 0.36
BRAF P15056 1/20 0.36
PBK Q96KB5 3/20 0.35
CYP3A4 P08684 1/20 0.34
ITGB3 P05106 1/20 0.33
ITGAV P06756 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21372781 0.91 IDO1 (0.42) IDO1TDO2BRAFPBKCYP3A4
SCHEMBL21372682 0.90 IDO1 (0.52) IDO1TDO2BRAF
SCHEMBL21372804 0.87 IDO1 (0.38) IDO1TDO2PBKCYP3A4
SCHEMBL21372664 0.86 ALDH1A1 (0.47) IDO1PBKCYP3A4
SCHEMBL21372902 0.86 IDO1 (0.46) IDO1TDO2HTR3EHTR3BHTR3A
SCHEMBL21372855 0.83 CYP3A4 (0.44) IDO1PBKCYP3A4
SCHEMBL21372864 0.82 CYP3A4 (0.38) PBKCYP3A4
SCHEMBL21373009 0.81 HTT (0.40) IDO1PBKCYP3A4
SCHEMBL21373044 0.81 MKNK1 (0.39) IDO1PBKCYP3A4
SCHEMBL21372715 0.81 IDO1 (0.46) IDO1TDO2BRAFPBKCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3294732-B1 BENZIMIDAZOLE AND IMADAZOPYRIDINE CARBOXIMIDAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF INDOLEAMINE 2,3-DIOXYGENASE GILEAD SCIENCES INC (US) 2019-09-25 EP claimed