SCHEMBL21386565

SCHEMBL21386565

Bc1ccc(-c2ccc(-c3ccc(-c4ccccc4)cc3F)c(F)c2F)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 4/20 0.39
HDAC6 Q9UBN7 2/20 0.38
ESR1 P03372 1/20 0.37
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
LMNA P02545 2/20 0.36
MAPT P10636 2/20 0.36
APAF1 O14727 1/20 0.36
NPC1 O15118 1/20 0.36
THRB P10828 1/20 0.36
XBP1 P17861 1/20 0.36
PTBP1 P26599 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
GALK1 P51570 1/20 0.36
BLM P54132 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19308568 0.91 DHODH (0.43) DHODHHDAC6ESR1ALOX5APFEN1
SCHEMBL23240088 0.90 FEN1 (0.42) HDAC6ESR1ALOX5APFEN1PDE3B
SCHEMBL19493701 0.90 PTGS1 (0.42) DHODHHDAC6ESR1ALOX5APFEN1
SCHEMBL23240031 0.88 FEN1 (0.44) DHODHHDAC6ESR1ALOX5APFEN1
SCHEMBL23510984 0.88 ALOX5AP (0.43) ALOX5APFEN1MEN1KMT2ALMNA
SCHEMBL23240080 0.86 MEN1 (0.40) DHODHHDAC6ESR1ALOX5APFEN1
SCHEMBL23240076 0.86 ALOX5AP (0.44) ALOX5APFEN1MEN1KMT2ALMNA
SCHEMBL19935706 0.83 DHODH (0.44) DHODHPDE3BPDE3AMEN1KMT2A
SCHEMBL19993178 0.82 ESR1 (0.38) ESR1ALOX5APFEN1PDE3BPDE3A
SCHEMBL20663902 0.82 MEN1 (0.48) DHODHESR1ALOX5APFEN1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022128845-A1 HETEROAROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2022-06-23 WO disclosed
WO-2022129018-A1 HETEROAROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2022-06-23 WO disclosed
WO-2022090099-A1 AROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2022-05-05 WO disclosed
WO-2021069535-A1 FLUORINATED AROMATIC COMPOUNDS MERCK PATENT GMBH (DE) 2021-04-15 WO disclosed
EP-3543313-B1 LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2020-10-07 EP disclosed
EP-3543314-A1 LIQUID-CRYSTALLINE MEDIUM Merck Patent GmbH (DE) 2019-09-25 EP disclosed