SCHEMBL21391013

SCHEMBL21391013

Cc1nc2ccc(C(C)(C)O)cc2n1C1(C)CCC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 2/20 0.42
PDE2A O00408 8/20 0.36
PDE10A Q9Y233 7/20 0.36
CYP11B1 P15538 2/20 0.36
CYP11B2 P19099 2/20 0.36
CCR5 P51681 1/20 0.35
ADRB1 P08588 1/20 0.34
ADRA2A P08913 1/20 0.34
CYP19A1 P11511 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
POLB P06746 1/20 0.32
APEX1 P27695 1/20 0.32
KARS1 Q15046 1/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
ACSS2 Q9NR19 2/20 0.31
ESRRA P11474 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21390825 0.79 HCAR1 (0.41) HCAR1PDE2APDE10ACYP11B1CYP11B2
SCHEMBL18779216 0.77 CSNK1D (0.39) POLBAPEX1KARS1
SCHEMBL21354649 0.77 RPS6KA3 (0.33) HCAR1PDE2APDE10APOLBAPEX1
SCHEMBL30315405 0.77 RPS6KA3 (0.33) HCAR1PDE2APDE10APOLBAPEX1
SCHEMBL21354651 0.77 RPS6KA3 (0.33) HCAR1PDE2APDE10APOLBAPEX1
SCHEMBL18779222 0.76 MCHR1 (0.35) HCAR1POLBAPEX1KARS1ESR1
SCHEMBL26008138 0.76 RPS6KA3 (0.33) HCAR1POLBAPEX1KARS1ESR1
SCHEMBL21375474 0.73 MCHR1 (0.33)
SCHEMBL21354650 0.73 MCHR1 (0.34) PDE2APDE10ACYP11B1CYP11B2ACSS2
SCHEMBL21375044 0.73 ALK (0.33) CCR5POLBAPEX1KARS1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183148-A1 KV7 CHANNEL ACTIVATORS COMPOSITIONS AND METHODS OF USE KNOPP BIOSCIENCES LLC (US) 2019-09-26 WO disclosed