SCHEMBL21397288

SCHEMBL21397288

C=CC(F)(F)c1cc(Cl)nnc1Cl

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.38
JUN P05412 1/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21397287 0.81 TDP1 (0.35) TDP1JUNNFKB1NFKB2RELA
SCHEMBL29708780 0.77 TDP1 (0.44) TDP1JUNNFKB1NFKB2RELA
SCHEMBL1204974 0.77 TDP1 (0.44) TDP1JUNNFKB1NFKB2RELA
SCHEMBL16701835 0.75 TDP1 (0.43) TDP1JUNNFKB1NFKB2RELA
SCHEMBL29899133 0.75 TDP1 (0.43) TDP1JUNNFKB1NFKB2RELA
SCHEMBL3075824 0.74 TDP1 (0.41) TDP1JUNNFKB1NFKB2RELA
SCHEMBL16701782 0.74 TDP1 (0.41) TDP1JUNNFKB1NFKB2RELA
SCHEMBL29919207 0.74 TDP1 (0.41) TDP1JUNNFKB1NFKB2RELA
SCHEMBL2424857 0.70 TDP1 (0.46) TDP1JUNNFKB1NFKB2RELA
SCHEMBL29417448 0.69 TDP1 (0.44) TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183367-A1 SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed