SCHEMBL21397537

SCHEMBL21397537

CC(C)(C)OC(=O)N1CCC2(CC1)Oc1ccccc1[C@H]2N

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.49
GPR119 Q8TDV5 3/20 0.45
KDM1A O60341 2/20 0.44
ABCB1 P08183 1/20 0.43
TSHR P16473 2/20 0.43
ALOX15 P16050 1/20 0.43
ATM Q13315 1/20 0.43
PTPN11 Q06124 4/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42
CHRM2 P08172 1/20 0.42
CHRM4 P08173 1/20 0.42
CHRM1 P11229 1/20 0.42
CHRM3 P20309 1/20 0.42
KDM4E B2RXH2 1/20 0.41
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2590439 0.86 GPR119 (0.42) IDO1GPR119KDM1ATSHRALOX15
SCHEMBL12541994 0.86 IDO1 (0.48) IDO1GPR119ABCB1TSHRALOX15
SCHEMBL15594335 0.84 MAPK1 (0.42) IDO1GPR119KDM1ATSHRALOX15
SCHEMBL23046063 0.83 IDO1 (0.50) IDO1GPR119KDM1AABCB1TSHR
SCHEMBL29890994 0.83 IDO1 (0.50) IDO1GPR119KDM1AABCB1TSHR
SCHEMBL22545150 0.81 POLB (0.47) GPR119PTPN11OPRD1OPRK1
SCHEMBL23169354 0.80 IDO1 (0.42) IDO1GPR119ABCB1TSHRALOX15
SCHEMBL12482111 0.80 IDO1 (0.58) IDO1GPR119ABCB1
SCHEMBL23500668 0.80 IDO1 (0.46) IDO1GPR119ABCB1TSHRALOX15
SCHEMBL23046236 0.80 IDO1 (0.46) IDO1GPR119ABCB1TSHRALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183367-A1 SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed