SCHEMBL2144010

SCHEMBL2144010

O=C(NO)c1cnc(N2C[C@]3(Cc4ccccc4)C[C@H]2CN3C(=O)O)nc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 20/20 0.48
HDAC1 Q13547 20/20 0.48
HDAC2 Q92769 20/20 0.48
HDAC6 Q9UBN7 20/20 0.48
HDAC4 P56524 15/20 0.48
HDAC7 Q8WUI4 15/20 0.48
HDAC10 Q969S8 15/20 0.48
HDAC11 Q96DB2 15/20 0.48
HDAC8 Q9BY41 15/20 0.48
HDAC9 Q9UKV0 15/20 0.48
HDAC5 Q9UQL6 15/20 0.48
CYP2D6 P10635 2/20 0.40
KCNH2 Q12809 1/20 0.40
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2145828 0.92 HDAC1 (0.45) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL1367543 0.81 HDAC6 (0.41) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL4539202 0.76 HDAC1 (0.60) HDAC1
SCHEMBL2143881 0.75 HDAC3 (0.40) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL1365585 0.73 HDAC6 (0.46) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL1365417 0.70 HDAC1 (0.57) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL12142364 0.68 HDAC1 (0.53) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL1366934 0.68 HDAC1 (0.53) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL4540562 0.68 HDAC1 (0.59) HDAC1
SCHEMBL7997961 0.67 HDAC6 (0.55) HDAC3HDAC1HDAC2HDAC6HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2489657-A2 Inhibitors of histone deacetylase MethylGene Inc. (CA) 2012-08-22 EP disclosed
EP-2343286-A1 Dibenzo[b,f][1,4]oxazepine derivatives as inhibitors of histone deacetylase Methylgene, Inc. (CA) 2011-07-13 EP disclosed