SCHEMBL21441968

SCHEMBL21441968

N#Cc1cc(F)c(-c2cnc(C(F)(F)F)nc2)cc1CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(F)cc1

nearest known ligand 0.65

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 19/20 0.65
ATM Q13315 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21716289 0.89 TRPA1 (0.78) TRPA1ATM
SCHEMBL18018197 0.89 TRPA1 (0.82) TRPA1
SCHEMBL16648077 0.89 TRPA1 (0.79) TRPA1
SCHEMBL18017576 0.85 TRPA1 (0.82) TRPA1
SCHEMBL16648243 0.84 TRPA1 (0.77) TRPA1
SCHEMBL20113258 0.83 TRPA1 (0.78) TRPA1
SCHEMBL18017805 0.83 TRPA1 (0.77) TRPA1ATM
SCHEMBL16648126 0.81 TRPA1 (0.79) TRPA1ATM
SCHEMBL16648093 0.81 TRPA1 (0.78) TRPA1
SCHEMBL18018379 0.81 TRPA1 (0.76) TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3256463-B1 1-(HET)ARYLSULFONYL-(PYRROLIDINE OR PIPERIDINE)-2-CARBOXAMIDE DERIVATIVES AND THEIR USE AS TRPA1 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2019-10-09 EP disclosed