SCHEMBL21443519

SCHEMBL21443519

CSc1ncc(C(N)=O)c(Oc2cccc(NC(=O)OC(C)(C)C)c2)n1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
NPSR1 Q6W5P4 3/20 0.52
KMT2A Q03164 3/20 0.52
ITK Q08881 2/20 0.49
MAPT P10636 1/20 0.49
HTT P42858 1/20 0.49
LMNA P02545 1/20 0.47
MAPK1 P28482 1/20 0.47
AURKA O14965 3/20 0.43
RPS6KB1 P23443 3/20 0.43
MEN1 O00255 2/20 0.42
SIRT2 Q8IXJ6 1/20 0.40
JAK2 O60674 1/20 0.40
SYK P43405 2/20 0.40
EGFR P00533 1/20 0.39
TDP2 O95551 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2362528 0.92 ALDH1A1 (0.54) ALDH1A1NPSR1KMT2AITKMAPT
SCHEMBL2288522 0.89 ALDH1A1 (0.57) ALDH1A1NPSR1KMT2AITKMAPT
SCHEMBL12518623 0.87 ALDH1A1 (0.70) ALDH1A1NPSR1KMT2AMAPTHTT
SCHEMBL21443465 0.86 ALDH1A1 (0.50) ALDH1A1NPSR1KMT2AITKMAPT
SCHEMBL21443521 0.84 ITK (0.49) ALDH1A1NPSR1KMT2AITKLMNA
SCHEMBL13498141 0.83 ALDH1A1 (0.52) ALDH1A1NPSR1KMT2AMAPTHTT
SCHEMBL12519591 0.82 ALDH1A1 (0.49) ALDH1A1NPSR1KMT2AMAPTHTT
SCHEMBL18720123 0.78 ITK (0.48) ALDH1A1NPSR1KMT2AITKMAPT
SCHEMBL13498135 0.77 SYK (0.55) ALDH1A1KMT2AITKMAPTHTT
SCHEMBL16670315 0.76 KMT2A (0.50) ALDH1A1NPSR1KMT2AMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3549934-A1 HETEROARYL COMPOUNDS AND USES THEREOF Celgene CAR LLC (BM) 2019-10-09 EP disclosed