SCHEMBL21443561

SCHEMBL21443561

Brc1coc([C@@H]2CCCNC2)n1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 3/20 0.39
CCNA2 P20248 3/20 0.39
CDK2 P24941 3/20 0.39
CCNA1 P78396 3/20 0.39
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
CDC7 O00311 1/20 0.36
PIM1 P11309 1/20 0.36
CSNK2B P67870 1/20 0.36
CSNK2A1 P68400 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13407530 0.81 HTR2A (0.39) CHEK1CCNA2CDK2CCNA1HTR2A
SCHEMBL3581077 0.73 MAPK11 (0.47) CHEK1CCNA2CDK2CCNA1HTR2A
SCHEMBL3581075 0.73 MAPK11 (0.47) CHEK1CCNA2CDK2CCNA1HTR2A
SCHEMBL3583291 0.71 ACP1 (0.41) CHEK1CCNA2CDK2CCNA1
SCHEMBL3583286 0.71 ACP1 (0.41) CHEK1CCNA2CDK2CCNA1
Hydrochloric Acid SCHEMBL4599388 0.70 ACP1 (0.40) CHEK1CCNA2CDK2CCNA1
SCHEMBL20028885 0.70 CHEK1 (0.43) CHEK1CCNA2CDK2CCNA1HTR2A
SCHEMBL3582287 0.70 MPO (0.40) CHEK1CCNA2CDK2CCNA1HTR2A
SCHEMBL3582283 0.70 MPO (0.40) CHEK1CCNA2CDK2CCNA1HTR2A
SCHEMBL30586799 0.70 NOTUM (0.39) CHEK1CCNA2CDK2CCNA1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3030233-B1 OXAZOLE OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME (US) 2019-10-09 EP disclosed