SCHEMBL21451900

SCHEMBL21451900

O=C1CCCCC1c1c(F)cccc1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR4 O00206 1/20 0.41
ABCB1 P08183 1/20 0.39
MCL1 Q07820 1/20 0.39
MAPT P10636 3/20 0.38
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
HCRTR1 O43613 2/20 0.36
HCRTR2 O43614 2/20 0.36
KMT2A Q03164 1/20 0.35
SCN9A Q15858 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34
DDB1 Q16531 1/20 0.34
CRBN Q96SW2 1/20 0.34
SLC18A3 Q16572 1/20 0.34
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21452202 0.87 TLR4 (0.40) TLR4MCL1MAPTCA1CA2
SCHEMBL16212320 0.86 ABCB1 (0.39) ABCB1MAPTCA1CA2HTR2C
SCHEMBL30496225 0.84 TP53 (0.43) TLR4MCL1MAPTCA1CA2
SCHEMBL21452414 0.84 TP53 (0.43) TLR4MCL1MAPTCA1CA2
SCHEMBL21452485 0.81 TLR4 (0.44) TLR4MCL1MAPTCA1CA2
SCHEMBL10356725 0.80 KDM4E (0.45) TLR4MCL1MAPTKMT2AALDH1A1
SCHEMBL21452480 0.76 P2RX7 (0.36) TLR4MCL1KDM4EHCAR1
SCHEMBL19993851 0.75 NPSR1 (0.40) TLR4MCL1MAPTCA1SCN9A
SCHEMBL1138365 0.74 KDM4E (0.47) TLR4HTR2CHTR2BKMT2ASLC18A3
SCHEMBL3228171 0.73 SLC6A4 (0.47) HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210171487-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF SHANGHAI JIANHE PHARMACEUTICAL & TECHNOLOGY CO. LTD. (CN) 2021-06-10 US disclosed
EP-3778579-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Jianhe Pharmaceutical & Technology Co. Ltd. (CN) 2021-02-17 EP disclosed
WO-2019192602-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海键合医药科技有限公司 2019-10-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210171487-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF CYP4F11, PAH, COMT TLR4 1217/4885ABCB1 167/4885MCL1 4533/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.