SCHEMBL21451901

SCHEMBL21451901

O=NC1(c2c(F)cccc2F)CCCCC1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 5/20 0.37
PDE7A Q13946 1/20 0.35
GRIN1 Q05586 3/20 0.32
GRIN2A Q12879 3/20 0.32
SLC6A4 P31645 2/20 0.32
GRIN2D O15399 2/20 0.32
GRIN3B O60391 2/20 0.32
GRIN2B Q13224 2/20 0.32
GRIN2C Q14957 2/20 0.32
GRIN3A Q8TCU5 2/20 0.32
LMNA P02545 2/20 0.32
OPRK1 P41145 1/20 0.32
OPRM1 P35372 1/20 0.32
CACNA1C Q13936 1/20 0.32
TNKS O95271 2/20 0.32
TNKS2 Q9H2K2 2/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HTT P42858 1/20 0.32
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21452518 0.87 HDAC4 (0.34) HDAC4
SCHEMBL21452575 0.85 TNKS (0.33) HDAC4TNKSTNKS2
SCHEMBL21451904 0.84 HDAC4 (0.48) HDAC4PDE7AGRIN1GRIN2ASLC6A4
SCHEMBL21452460 0.76 GRIN1 (0.45) HDAC4PDE7AGRIN1GRIN2ASLC6A4
SCHEMBL21452462 0.74 PDE7A (0.37) PDE7AGRIN1GRIN2ASLC6A4GRIN2D
SCHEMBL21452512 0.74 PDE7A (0.40) HDAC4PDE7AGRIN1GRIN2ASLC6A4
SCHEMBL21452501 0.73 PDE7A (0.36) PDE7AGRIN1GRIN2ASLC6A4GRIN2D
SCHEMBL21452174 0.72 HDAC4 (0.39) HDAC4PDE7AGRIN1GRIN2ASLC6A4
SCHEMBL21452189 0.72 SLC6A4 (0.47) SLC6A4OPRK1OPRM1
SCHEMBL21452484 0.72 HDAC4 (0.36) HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3778579-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Jianhe Pharmaceutical & Technology Co. Ltd. (CN) 2021-02-17 EP disclosed
WO-2019192602-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海键合医药科技有限公司 2019-10-10 WO disclosed