SCHEMBL2146325

SCHEMBL2146325

CC(C)(C)OC(=O)C1(F)CCN(Cc2ccccc2)C1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 13/20 0.49
CYP3A4 P08684 9/20 0.49
TSHR P16473 5/20 0.49
NPFFR1 Q9GZQ6 1/20 0.47
NPFFR2 Q9Y5X5 1/20 0.47
P4HB P07237 1/20 0.46
CYP1A2 P05177 4/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
ALDH1A1 P00352 3/20 0.45
HPGD P15428 1/20 0.44
USP2 O75604 3/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14962729 0.86 CYP2D6 (0.53) CYP2D6CYP3A4TSHRCYP1A2CYP2C9
SCHEMBL14962728 0.86 CYP2D6 (0.53) CYP2D6CYP3A4TSHRCYP1A2CYP2C9
SCHEMBL14677254 0.86 CYP2D6 (0.53) CYP2D6CYP3A4TSHRCYP1A2CYP2C9
SCHEMBL14957149 0.81 CYP2D6 (0.54) CYP2D6CYP3A4TSHRCYP1A2CYP2C9
SCHEMBL14957312 0.81 CYP2D6 (0.54) CYP2D6CYP3A4TSHRCYP1A2CYP2C9
SCHEMBL14965694 0.81 CYP2D6 (0.54) CYP2D6CYP3A4TSHRCYP1A2CYP2C9
SCHEMBL31334693 0.81 NPFFR1 (0.53) CYP2D6CYP3A4TSHRNPFFR1NPFFR2
SCHEMBL2158292 0.81 DRD2 (0.53) CYP2D6CYP3A4TSHRNPFFR1NPFFR2
SCHEMBL21262272 0.79 CYP2D6 (0.60) CYP2D6CYP3A4TSHRCYP1A2CYP2C9
SCHEMBL1426231 0.78 CYP2D6 (0.64) CYP2D6CYP3A4TSHRCYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011088045-A1 AURORA KINASE COMPOUNDS AND METHODS OF THEIR USE AMBIT BIOSCIENCES CORPORATION (US) 2011-07-21 WO disclosed