SCHEMBL21470159

SCHEMBL21470159

C/C(=C\c1ccc(Cl)c(C(F)(F)F)c1)C(=O)Nc1ccccc1C(=O)O

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 4/20 0.64
TRPM8 Q7Z2W7 2/20 0.64
CLCN2 P51788 1/20 0.49
TRPA1 O75762 3/20 0.46
GRIK1 P39086 2/20 0.46
TAS2R14 Q9NYV8 4/20 0.44
ALDH1A1 P00352 4/20 0.44
MAPT P10636 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
KDM4E B2RXH2 2/20 0.44
NPC1 O15118 1/20 0.44
NFKB1 P19838 1/20 0.44
RAB9A P51151 1/20 0.44
GFER P55789 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PPARG P37231 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8048240 0.87 DHODH (0.71) DHODHTRPM8CLCN2TRPA1ALDH1A1
SCHEMBL8048243 0.87 DHODH (0.71) DHODHTRPM8CLCN2TRPA1ALDH1A1
SCHEMBL21470162 0.83 DHODH (0.68) DHODHTRPM8TRPA1ALDH1A1MAPT
SCHEMBL8048868 0.82 TRPM8 (0.76) DHODHTRPM8TRPA1GRIK1TAS2R14
SCHEMBL8048873 0.82 TRPM8 (0.76) DHODHTRPM8TRPA1GRIK1TAS2R14
SCHEMBL29966740 0.82 TRPM8 (0.76) DHODHTRPM8TRPA1GRIK1TAS2R14
SCHEMBL8060484 0.82 DHODH (0.70) DHODHTRPM8TRPA1GRIK1TAS2R14
SCHEMBL8060487 0.82 DHODH (0.70) DHODHTRPM8TRPA1GRIK1TAS2R14
SCHEMBL8060378 0.81 TRPM8 (0.74) DHODHTRPM8TRPA1GRIK1TAS2R14
Lithium SCHEMBL8048874 0.81 TRPM8 (0.74) DHODHTRPM8TRPA1GRIK1TAS2R14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019196714-A1 N-SUBSTITUTED ACRYLAMIDE DERIVATIVE AS DHODH INHIBITOR, AND PREPARATION AND USE THEREOF 华东理工大学 2019-10-17 WO disclosed