SCHEMBL21470195

SCHEMBL21470195

C/C(=C\c1ccc(-c2ccccc2)cc1)C(=O)Nc1ccccc1C(=O)O

nearest known ligand 0.84

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 3/20 0.84
TRPM8 Q7Z2W7 2/20 0.84
TRPM2 O94759 5/20 0.59
LTB4R Q15722 1/20 0.59
TRPA1 O75762 5/20 0.57
PTPN1 P18031 1/20 0.50
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.45
MAPT P10636 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C19 P33261 1/20 0.45
SUCNR1 Q9BXA5 1/20 0.45
STAT1 P42224 2/20 0.45
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8065734 0.91 DHODH (1.00) DHODHTRPM8TRPM2LTB4RTRPA1
SCHEMBL8065731 0.91 DHODH (1.00) DHODHTRPM8TRPM2LTB4RTRPA1
SCHEMBL8061709 0.89 DHODH (0.84) DHODHTRPM8TRPM2LTB4RTRPA1
SCHEMBL8141640 0.89 DHODH (0.84) DHODHTRPM8TRPM2LTB4RTRPA1
SCHEMBL8061707 0.89 DHODH (0.84) DHODHTRPM8TRPM2LTB4RTRPA1
SCHEMBL8141637 0.89 DHODH (0.84) DHODHTRPM8TRPM2LTB4RTRPA1
SCHEMBL8049316 0.88 DHODH (0.82) DHODHTRPM8TRPM2LTB4RTRPA1
SCHEMBL8049318 0.88 DHODH (0.82) DHODHTRPM8TRPM2LTB4RTRPA1
SCHEMBL8061608 0.88 DHODH (0.82) DHODHTRPM8TRPM2LTB4RTRPA1
SCHEMBL8061602 0.88 DHODH (0.82) DHODHTRPM8TRPM2LTB4RTRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019196714-A1 N-SUBSTITUTED ACRYLAMIDE DERIVATIVE AS DHODH INHIBITOR, AND PREPARATION AND USE THEREOF 华东理工大学 2019-10-17 WO disclosed