SCHEMBL21473350

SCHEMBL21473350

COc1ccc(C(OCC2CCC(n3cc(C)c(NC(=O)c4ccccc4)nc3=O)O2)(c2ccccc2)c2ccc(OC)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.47
RIN1 Q13671 1/20 0.47
TMIGD3 P0DMS9 4/20 0.39
ADORA3 P0DMS8 11/20 0.39
ADORA1 P30542 2/20 0.39
TYMP P19971 1/20 0.38
ADORA2A P29274 2/20 0.37
SLC6A1 P30531 2/20 0.37
SLC6A11 P48066 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
ADORA2B P29275 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26190472 1.00 ABL1 (0.47) ABL1RIN1TMIGD3ADORA3ADORA1
SCHEMBL22984016 0.87 TYMP (0.46) TMIGD3ADORA3ADORA1TYMP
SCHEMBL21828786 0.87 TYMP (0.46) TMIGD3ADORA3ADORA1TYMP
SCHEMBL261967 0.87 TYMP (0.46) TMIGD3ADORA3ADORA1TYMP
SCHEMBL23056605 0.86 ABL1 (0.65) ABL1RIN1ADORA3TYMPADORA2A
SCHEMBL21504687 0.86 POLB (0.40) ABL1RIN1TMIGD3ADORA3ADORA1
SCHEMBL3070618 0.83 TYMP (0.54) TYMP
SCHEMBL3070612 0.83 TYMP (0.54) TYMP
SCHEMBL22983996 0.83 POLB (0.40) ABL1RIN1TMIGD3ADORA3ADORA1
SCHEMBL31725429 0.83 TYMP (0.39) ABL1RIN1TMIGD3ADORA3ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019200273-A1 NOVEL PHOSPHOROUS (V)-BASED REAGENTS, PROCESSES FOR THE PREPARATION THEREOF, AND THEIR USE IN MAKING STEREO-DEFINED ORGANOPHOSHOROUS (V) COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2019-10-17 WO disclosed