SCHEMBL21473594

SCHEMBL21473594

C[C@@H](c1ccccc1)c1nc2ccccc2s1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.65
LOXL2 Q9Y4K0 1/20 0.58
CASR P41180 1/20 0.57
MAPK1 P28482 2/20 0.50
TSHR P16473 2/20 0.50
ALOX5 P09917 1/20 0.50
GAA P10253 1/20 0.50
RAB9A P51151 3/20 0.49
MAPT P10636 1/20 0.49
PAX8 Q06710 1/20 0.49
NOD2 Q9HC29 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
KMT2A Q03164 1/20 0.49
HSD17B10 Q99714 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
HIF1A Q16665 1/20 0.48
ALDH1A1 P00352 2/20 0.44
CSNK1D P48730 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22997080 1.00 HPGD (0.65) HPGDLOXL2CASRMAPK1TSHR
SCHEMBL2146969 0.89 LOXL2 (0.66) HPGDLOXL2CASRMAPK1TSHR
SCHEMBL29449586 0.83 HPGD (0.58) HPGDLOXL2CASRMAPK1TSHR
SCHEMBL29449578 0.83 HPGD (0.58) HPGDLOXL2CASRMAPK1TSHR
SCHEMBL5851278 0.81 HPGD (0.69) HPGDLOXL2CASRMAPK1TSHR
SCHEMBL62420 0.81 LOXL2 (0.66) HPGDLOXL2CASRMAPK1TSHR
SCHEMBL10857871 0.80 HPGD (0.67) HPGDLOXL2CASRMAPK1TSHR
SCHEMBL5560135 0.80 CASR (0.49) HPGDLOXL2CASRMAPK1TSHR
SCHEMBL9675088 0.79 LOXL2 (0.64) HPGDLOXL2CASRMAPK1TSHR
SCHEMBL900511 0.79 HPGD (1.00) HPGDLOXL2CASRMAPK1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019196938-A1 QUINAZOLINE COMPOUND SERVING AS EGFR TRIPLE MUTATION INHIBITOR AND APPLICATIONS THEREOF 华东理工大学 2019-10-17 WO disclosed