SCHEMBL21476667

SCHEMBL21476667

COC(=O)CCc1cncc(-c2c(C)cccc2OC)c1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSA P10619 3/20 0.43
FFAR1 O14842 7/20 0.42
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
CNR2 P34972 1/20 0.41
KCNH2 Q12809 1/20 0.40
HDAC1 Q13547 1/20 0.39
VDR P11473 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21475993 0.92 FFAR1 (0.48) FFAR1CYP11B1CYP11B2CNR2HDAC1
SCHEMBL21476085 0.87 CYP11B1 (0.41) CTSAFFAR1CYP11B1CYP11B2CNR2
SCHEMBL21475921 0.82 CYP11B1 (0.42) FFAR1CYP11B1CYP11B2CNR2HDAC1
SCHEMBL31303333 0.78 CTSA (0.54) CTSA
SCHEMBL21459985 0.78 CTSA (0.54) CTSA
SCHEMBL21459983 0.78 CTSA (0.54) CTSA
SCHEMBL21475996 0.77 FFAR1 (0.64) FFAR1
SCHEMBL21476056 0.77 FFAR1 (0.52) FFAR1
SCHEMBL21476702 0.76 FFAR1 (0.66) FFAR1SIRT2
SCHEMBL3745313 0.73 CYP11B2 (0.48) CTSAFFAR1CYP11B1CYP11B2CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019200202-A1 ANTAGONISTS OF HUMAN INTEGRIN (ALPHA4)(BETA7) MORPHIC THERAPEUTIC, INC. (US) 2019-10-17 WO disclosed