SCHEMBL21481599

SCHEMBL21481599

C=C1CCC(Cn2ncc3c(N)nc(Cl)nc32)CC1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.39
ADORA1 P30542 1/20 0.39
NT5E P21589 2/20 0.34
PKM P14618 1/20 0.33
PDE1A P54750 1/20 0.32
PDE1B Q01064 1/20 0.32
PDE1C Q14123 1/20 0.32
CYP3A4 P08684 4/20 0.31
CYP2D6 P10635 2/20 0.31
MERTK Q12866 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21481598 0.84 ADORA2A (0.39) ADORA2AADORA1NT5EPKMPDE1A
SCHEMBL30095986 0.76 ADORA2A (0.39) ADORA2AADORA1PDE1APDE1BPDE1C
SCHEMBL21462258 0.75 CYP3A4 (0.39) ADORA2AADORA1CYP3A4CYP2D6MERTK
SCHEMBL30748227 0.73 ADORA2A (0.38) ADORA2AADORA1PKMPDE1APDE1B
SCHEMBL29174854 0.73 ADORA2A (0.38) ADORA2AADORA1PKMPDE1APDE1B
SCHEMBL25876067 0.73 PDE1A (0.41) ADORA2AADORA1PDE1APDE1BPDE1C
SCHEMBL21481606 0.68 ADORA2A (0.52) ADORA2AADORA1PKMCYP3A4CYP2D6
SCHEMBL31385338 0.68 ADORA2A (0.52) ADORA2AADORA1PKMCYP3A4CYP2D6
SCHEMBL21481670 0.67 KDM4E (0.46) ADORA2AADORA1CYP3A4CYP2D6
SCHEMBL21462235 0.66 CYP3A4 (0.64) PKMCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019196918-A1 FIVE-MEMBERED HETEROCYCLO-PYRIMIDINE COMPOUND, PHARMACEUTICAL COMPOSITION AND USE THEREOF 罗欣药业(上海)有限公司 2019-10-17 WO disclosed