SCHEMBL21481598

SCHEMBL21481598

Nc1nc(Cl)nc2c1cnn2CC1CCC(CBr)CC1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.39
ADORA1 P30542 1/20 0.39
NT5E P21589 2/20 0.34
ALDH1A1 P00352 2/20 0.34
ALDH1A2 O94788 1/20 0.34
ALDH1A3 P47895 1/20 0.34
PKM P14618 1/20 0.33
MERTK Q12866 4/20 0.33
PDE1A P54750 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE1C Q14123 1/20 0.33
HSP90AA1 P07900 2/20 0.32
TRAP1 Q12931 2/20 0.32
HSP90AB1 P08238 1/20 0.32
HTT P42858 1/20 0.32
CYP3A4 P08684 3/20 0.32
HSP90B1 P14625 1/20 0.32
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21481599 0.84 ADORA2A (0.39) ADORA2AADORA1NT5EPKMMERTK
SCHEMBL30095986 0.79 ADORA2A (0.39) ADORA2AADORA1ALDH1A1ALDH1A2ALDH1A3
SCHEMBL25876067 0.77 PDE1A (0.41) ADORA2AADORA1ALDH1A1ALDH1A2ALDH1A3
SCHEMBL30748227 0.77 ADORA2A (0.38) ADORA2AADORA1ALDH1A1ALDH1A2ALDH1A3
SCHEMBL29174854 0.77 ADORA2A (0.38) ADORA2AADORA1ALDH1A1ALDH1A2ALDH1A3
SCHEMBL21465889 0.75 CYP3A4 (0.40) ADORA2AADORA1ALDH1A1ALDH1A2ALDH1A3
SCHEMBL21462262 0.75 CYP3A4 (0.40) ADORA2AADORA1ALDH1A1ALDH1A2ALDH1A3
SCHEMBL21481752 0.75 CYP3A4 (0.40) ADORA2AADORA1ALDH1A1ALDH1A2ALDH1A3
SCHEMBL21465886 0.75 TLR7 (0.46) ADORA2AADORA1MERTKPDE1APDE1B
SCHEMBL28651973 0.69 GRM2 (0.34) ADORA2AADORA1PKMMERTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019196918-A1 FIVE-MEMBERED HETEROCYCLO-PYRIMIDINE COMPOUND, PHARMACEUTICAL COMPOSITION AND USE THEREOF 罗欣药业(上海)有限公司 2019-10-17 WO disclosed