SCHEMBL21484083

SCHEMBL21484083

CC(C)c1cnn2c(NCc3ccccc3-c3ccc4ccccc4n3)nc(N3CCC(NC(=O)OCc4ccccc4)CC3)nc12

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 14/20 0.42
CDK9 P50750 13/20 0.42
CCNE1 P24864 2/20 0.39
SMPD3 Q9NY59 1/20 0.37
CDK5 Q00535 2/20 0.37
CDK5R1 Q15078 2/20 0.37
CCNT1 O60563 1/20 0.37
CCNA2 P20248 1/20 0.37
CDK7 P50613 1/20 0.37
CCNH P51946 1/20 0.37
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
CSNK1A1 P48729 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23381749 0.83 CDK9 (0.46) CDK2CDK9CCNE1CDK5CDK5R1
SCHEMBL23382180 0.82 CDK9 (0.45) CDK2CDK9CCNE1CDK5CDK5R1
SCHEMBL23382008 0.80 CDK9 (0.42) CDK2CDK9CCNE1CDK5CDK5R1
SCHEMBL23382145 0.79 CNR1 (0.44) CDK2CDK9SMPD3CNR1CNR2
SCHEMBL23382029 0.78 CDK9 (0.41) CDK2CDK9CCNE1CDK5CDK5R1
SCHEMBL23382112 0.77 CKS1B (0.41) CDK2CDK9CCNE1CDK5CDK7
SCHEMBL23381671 0.77 CDK2 (0.56) CDK2CDK9CCNE1CDK5CDK5R1
SCHEMBL23381992 0.75 CDK9 (0.51) CDK2CDK9CCNE1CDK5CDK5R1
SCHEMBL23381996 0.75 CDK9 (0.51) CDK2CDK9CCNE1CDK5CDK5R1
SCHEMBL23382195 0.75 CDK9 (0.51) CDK2CDK9CCNE1CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019197549-A1 PYRAZOLO-TRIAZINE AND/OR PYRAZOLO-PYRIMIDINE DERIVATIVES AS SELECTIVE INHIBITOR OF CYCLIN DEPENDENT KINASE QURIENT CO., LTD. (KR) 2019-10-17 WO disclosed