SCHEMBL2148586

SCHEMBL2148586

CCc1cc(Nc2nc(Sc3ccc(N)cc3)nc3cccn23)n[nH]1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AURKA O14965 17/20 0.36
AURKB Q96GD4 16/20 0.36
GSK3B P49841 4/20 0.36
SRC P12931 3/20 0.36
NTRK1 P04629 1/20 0.34
AURKC Q9UQB9 1/20 0.34
ABL1 P00519 1/20 0.33
BCR P11274 1/20 0.33
GRK6 P43250 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2148867 0.89 AURKA (0.47) AURKAAURKBGSK3BSRCNTRK1
SCHEMBL2169274 0.84 AURKB (0.47) AURKAAURKBGSK3BSRCAURKC
SCHEMBL2149092 0.82 AURKA (0.32) AURKAAURKBGSK3BSRCNTRK1
SCHEMBL2148630 0.82 AURKA (0.32) AURKAAURKBGSK3BSRCNTRK1
SCHEMBL2153217 0.81 SRC (0.44) AURKAAURKBGSK3BSRCNTRK1
SCHEMBL2203289 0.80 AURKA (0.47) AURKAAURKBGSK3BSRCNTRK1
SCHEMBL2169069 0.79 GRK6 (0.39) AURKANTRK1GRK6
SCHEMBL2159843 0.77 AURKA (0.43) AURKAAURKBGSK3BSRCNTRK1
SCHEMBL2149892 0.76 AURKA (0.61) AURKAAURKBAURKC
SCHEMBL2948567 0.75 AURKB (0.64) AURKAAURKBGSK3BSRCAURKC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011088045-A1 AURORA KINASE COMPOUNDS AND METHODS OF THEIR USE AMBIT BIOSCIENCES CORPORATION (US) 2011-07-21 WO disclosed