SCHEMBL2148749

SCHEMBL2148749

O=C(O)N1CC(O)C(c2ccc(F)cc2)C1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TLR2 O60603 1/20 0.41
TLR1 Q15399 1/20 0.41
SLC6A3 Q01959 2/20 0.40
SLC6A4 P31645 1/20 0.40
HRH3 Q9Y5N1 2/20 0.40
KDM1A O60341 2/20 0.39
SLC9A1 P19634 1/20 0.39
ALDH1A1 P00352 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
ATM Q13315 1/20 0.38
MYC P01106 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
PAX8 Q06710 1/20 0.38
MAPT P10636 1/20 0.37
TACR1 P25103 1/20 0.37
SLC18A3 Q16572 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6041432 0.86 RAB9A (0.45) HRH3ALDH1A1NPC1RAB9AATM
SCHEMBL5200432 0.86 RAB9A (0.45) TLR2TLR1HRH3ALDH1A1NPC1
SCHEMBL4328689 0.86 RAB9A (0.45) TLR2TLR1HRH3ALDH1A1NPC1
SCHEMBL27708147 0.86 RAB9A (0.45) TLR2TLR1HRH3ALDH1A1NPC1
SCHEMBL23923863 0.84 MYC (0.49) TLR2TLR1SLC6A3SLC6A4HRH3
SCHEMBL6127033 0.84 MYC (0.49) TLR2TLR1SLC6A3SLC6A4HRH3
SCHEMBL6127038 0.84 MYC (0.49) TLR2TLR1SLC6A3SLC6A4HRH3
SCHEMBL17514137 0.83 CYP1A2 (0.43) TLR2TLR1NPC1RAB9AMAPT
SCHEMBL23924236 0.82 TLR2 (0.46) TLR2TLR1SLC6A3HRH3KDM1A
SCHEMBL15397583 0.82 KDM1A (0.50) TLR2TLR1SLC6A3SLC6A4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011088045-A1 AURORA KINASE COMPOUNDS AND METHODS OF THEIR USE AMBIT BIOSCIENCES CORPORATION (US) 2011-07-21 WO disclosed