SCHEMBL21495095

SCHEMBL21495095

O=C[C@@H](Br)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
AHR P35869 2/20 0.41
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37
IDO2 Q6ZQW0 1/20 0.37
TP53 P04637 1/20 0.36
CYP1B1 Q16678 1/20 0.35
MAPK1 P28482 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
SLC6A3 Q01959 7/20 0.35
SLC6A2 P23975 6/20 0.35
SLC6A4 P31645 6/20 0.35
KCNH2 Q12809 4/20 0.35
CYP3A4 P08684 4/20 0.35
CYP2D6 P10635 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL747175 1.00 ALDH1A1 (0.43) ALDH1A1AHRLMNAHTTSMN1; SMN2
SCHEMBL12615184 0.84 SLC6A2 (0.40) ALDH1A1LMNAHTTSMN1; SMN2SLC6A3
SCHEMBL26968200 0.84 S1PR1 (0.33) ALDH1A1
SCHEMBL3973135 0.82 PSEN1 (0.35) ALDH1A1SLC6A3SLC6A2SLC6A4KCNH2
SCHEMBL4621988 0.82 S1PR1 (0.38) ALDH1A1SMN1; SMN2MAPK1SLC6A3
SCHEMBL20722071 0.82 PSEN1 (0.35) ALDH1A1SLC6A3SLC6A2SLC6A4KCNH2
SCHEMBL1701138 0.82 MDM2 (0.40) ALDH1A1HTTSLC6A3SLC6A2SLC6A4
SCHEMBL2550930 0.78 ALDH1A1 (0.46) ALDH1A1AHRLMNAHTTSMN1; SMN2
SCHEMBL20551343 0.78 KDR (0.41) IDO1SLC6A3
SCHEMBL1726228 0.78 KDR (0.41) IDO1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3997096-A1 NEW HETEROCYCLIC COMPOUNDS F. Hoffmann-La Roche AG (CH) 2022-05-18 EP disclosed
WO-2021005034-A1 NEW HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2021-01-14 WO disclosed
WO-2019201867-A1 SUBSTITUTED PROPANAMIDES AS INHIBITORS OF NUCLEASES MASARYKOVA UNIVERZITA (CZ) 2019-10-24 WO disclosed